Literature DB >> 1404240

Fatty acid amides: scooting mode-based discovery of tight-binding competitive inhibitors of secreted phospholipases A2.

M K Jain1, F Ghomashchi, B Z Yu, T Bayburt, D Murphy, D Houck, J Brownell, J C Reid, J E Solowiej, S M Wong.   

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Year:  1992        PMID： 1404240     DOI： 10.1021/jm00097a018

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  8 in total

1.  One pot direct synthesis of amides or oxazolines from carboxylic acids using Deoxo-Fluor reagent.

Authors:  Cyrous O Kangani; David E Kelley
Journal:  Tetrahedron Lett       Date:  2005-12-19       Impact factor: 2.415

Review 2.  Phospholipase A2 enzymes: physical structure, biological function, disease implication, chemical inhibition, and therapeutic intervention.

Authors:  Edward A Dennis; Jian Cao; Yuan-Hao Hsu; Victoria Magrioti; George Kokotos
Journal:  Chem Rev       Date:  2011-09-12       Impact factor: 60.622

3.  Chemical requirements for inhibition of gap junction communication by the biologically active lipid oleamide.

Authors:  D L Boger; J E Patterson; X Guan; B F Cravatt; R A Lerner; N B Gilula
Journal:  Proc Natl Acad Sci U S A       Date:  1998-04-28       Impact factor: 11.205

4.  Structural requirements for 5-HT2A and 5-HT1A serotonin receptor potentiation by the biologically active lipid oleamide.

Authors:  D L Boger; J E Patterson; Q Jin
Journal:  Proc Natl Acad Sci U S A       Date:  1998-04-14       Impact factor: 11.205

5.  Primary fatty acid amide metabolism: conversion of fatty acids and an ethanolamine in N18TG2 and SCP cells.

Authors:  Emma K Farrell; Yuden Chen; Muna Barazanji; Kristen A Jeffries; Felipe Cameroamortegui; David J Merkler
Journal:  J Lipid Res       Date:  2011-11-16       Impact factor: 5.922

6.  Erucamide as a modulator of water balance: new function of a fatty acid amide.

Authors:  Anders Hamberger; Gunnar Stenhagen
Journal:  Neurochem Res       Date:  2003-02       Impact factor: 3.996

7.  Structure-based design of the first potent and selective inhibitor of human non-pancreatic secretory phospholipase A2.

Authors:  R W Schevitz; N J Bach; D G Carlson; N Y Chirgadze; D K Clawson; R D Dillard; S E Draheim; L W Hartley; N D Jones; E D Mihelich
Journal:  Nat Struct Biol       Date:  1995-06

Review 8.  pCRP-mCRP Dissociation Mechanisms as Potential Targets for the Development of Small-Molecule Anti-Inflammatory Chemotherapeutics.

Authors:  Vittorio Caprio; Lina Badimon; Mario Di Napoli; Wen-Hui Fang; Glenn R Ferris; Baoqiang Guo; Rocco S Iemma; Donghui Liu; Yasmin Zeinolabediny; Mark Slevin
Journal:  Front Immunol       Date:  2018-05-28       Impact factor: 7.561
  8 in total

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