Literature DB >> 1333459

A simple synthesis of [11C]methyl triflate.

D M Jewett1.   

Abstract

[11C]Methyl triflate ([11C]methyl trifluoromethanesulfonate) was formed in high yield when [11C]methyl iodide in a nitrogen carrier was passed at 200 degrees C through a column containing graphitized carbon impregnated with 50% by weight of silver triflate.

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Year:  1992        PMID: 1333459     DOI: 10.1016/0883-2889(92)90012-4

Source DB:  PubMed          Journal:  Int J Rad Appl Instrum A        ISSN: 0883-2889


  36 in total

1.  Development and optimization of a novel automated loop method for production of [11C]nicotine.

Authors:  Arijit Ghosh; Karen Woolum; Michael V Knopp; Krishan Kumar
Journal:  Appl Radiat Isot       Date:  2018-05-30       Impact factor: 1.513

2.  Analogs of JHU75528, a PET ligand for imaging of cerebral cannabinoid receptors (CB1): development of ligands with optimized lipophilicity and binding affinity.

Authors:  Hong Fan; Evangelia Kotsikorou; Alexander F Hoffman; Hayden T Ravert; Daniel Holt; Dow P Hurst; Carl R Lupica; Patricia H Reggio; Robert F Dannals; Andrew G Horti
Journal:  Eur J Med Chem       Date:  2008-04-18       Impact factor: 6.514

3.  Synthesis and in vivo evaluation of [11C]tariquidar, a positron emission tomography radiotracer based on a third-generation P-glycoprotein inhibitor.

Authors:  Florian Bauer; Claudia Kuntner; Jens P Bankstahl; Thomas Wanek; Marion Bankstahl; Johann Stanek; Severin Mairinger; Bernd Dörner; Wolfgang Löscher; Markus Müller; Thomas Erker; Oliver Langer
Journal:  Bioorg Med Chem       Date:  2010-06-22       Impact factor: 3.641

4.  Synthesis and in vivo brain distribution of carbon-11-labeled δ-opioid receptor agonists.

Authors:  Rama Pichika; Douglas M Jewett; Philip S Sherman; John R Traynor; Stephen M Husbands; James H Woods; Michael R Kilbourn
Journal:  Nucl Med Biol       Date:  2010-07-24       Impact factor: 2.408

Review 5.  Considerations in the Development of Reversibly Binding PET Radioligands for Brain Imaging.

Authors:  Victor W Pike
Journal:  Curr Med Chem       Date:  2016       Impact factor: 4.530

6.  Translocator protein ligands based on N-methyl-(quinolin-4-yl)oxypropanamides with properties suitable for PET radioligand development.

Authors:  Chad Brouwer; Kimberly J Jenko; Sami S Zoghbi; Cheryl L Morse; Robert B Innis; Victor W Pike
Journal:  Eur J Med Chem       Date:  2016-08-25       Impact factor: 6.514

7.  Rapid Room-Temperature 11C-Methylation of Arylamines with [11C]Methyl Iodide Promoted by Solid Inorganic Bases in DMF.

Authors:  Lisheng Cai; Rong Xu; Xuelei Guo; Victor W Pike
Journal:  European J Org Chem       Date:  2012-03

8.  Synthesis and small-animal positron emission tomography evaluation of [11C]-elacridar as a radiotracer to assess the distribution of P-glycoprotein at the blood-brain barrier.

Authors:  Bernd Dörner; Claudia Kuntner; Jens P Bankstahl; Marion Bankstahl; Johann Stanek; Thomas Wanek; Gloria Stundner; Severin Mairinger; Wolfgang Löscher; Markus Müller; Oliver Langer; Thomas Erker
Journal:  J Med Chem       Date:  2009-10-08       Impact factor: 7.446

9.  Fully automated synthesis and initial PET evaluation of [11C]PBR28.

Authors:  Min Wang; Karmen K Yoder; Mingzhang Gao; Bruce H Mock; Xiao-Ming Xu; Andrew J Saykin; Gary D Hutchins; Qi-Huang Zheng
Journal:  Bioorg Med Chem Lett       Date:  2009-08-15       Impact factor: 2.823

10.  Test-retest variability of quantitative [11C]PIB studies in Alzheimer's disease.

Authors:  Nelleke Tolboom; Maqsood Yaqub; Ronald Boellaard; Gert Luurtsema; Albert D Windhorst; Philip Scheltens; Adriaan A Lammertsma; Bart N M van Berckel
Journal:  Eur J Nucl Med Mol Imaging       Date:  2009-04-22       Impact factor: 9.236

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