Literature DB >> 12824041

Synthesis and structure-activity relationships of open D-Ring galanthamine analogues.

Denyse Herlem1, Marie Thérèse Martin, Claude Thal, Catherine Guillou.   

Abstract

Open D-ring galanthamine analogues were prepared using ring-opening reactions of the quaternarized urethane or oxazolidine functions and were evaluated for their acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) inhibition potency.

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Year:  2003        PMID： 12824041     DOI： 10.1016/s0960-894x(03)00397-4

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  3 in total

1.  Electronic structure and PCA analysis of covalent and non-covalent acetylcholinesterase inhibitors.

Authors:  Erica Cristina Moreno Nascimento; João B L Martins
Journal:  J Mol Model       Date:  2010-09-14       Impact factor: 1.810

2.  Quantification of Galantamine in Sternbergia Species by High Performance Liquid Chromatography.

Authors:  Özlem Bahadır Acikara; Betül Sever Yilmaz; Dilhun Yazgan; Gülçin Saltan Işcan
Journal:  Turk J Pharm Sci       Date:  2018-12-31

3.  Galantamine-Curcumin Hybrids as Dual-Site Binding Acetylcholinesterase Inhibitors.

Authors:  Georgi Stavrakov; Irena Philipova; Atanas Lukarski; Mariyana Atanasova; Dimitrina Zheleva; Zvetanka D Zhivkova; Stefan Ivanov; Teodora Atanasova; Spiro Konstantinov; Irini Doytchinova
Journal:  Molecules       Date:  2020-07-23       Impact factor: 4.411
  3 in total

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