Literature DB >> 12667692

Effects of a series of dihydroanthracene derivatives on drug efflux in multidrug resistant cancer cells.

Sandrine Alibert1, Christiane Santelli-Rouvier, Madeleine Castaing, Michel Berthelot, Gabriella Spengler, Jozsef Molnar, Jacques Barbe.   

Abstract

A set of 9,10-dihydro-9,10-ethano and ethenoanthracene derivatives was tested with the aim to quantify the effect observed on drug efflux. Structure activity relationships and molecular modeling studies allowed to define topological display of pharmacophoric groups for these reversal agents.

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Year:  2003        PMID: 12667692     DOI: 10.1016/s0223-5234(03)00018-7

Source DB:  PubMed          Journal:  Eur J Med Chem        ISSN: 0223-5234            Impact factor:   6.514


  3 in total

1.  Design, Synthesis and Biochemical Evaluation of Novel Ethanoanthracenes and Related Compounds to Target Burkitt's Lymphoma.

Authors:  Andrew J Byrne; Sandra A Bright; James P McKeown; John E O'Brien; Brendan Twamley; Darren Fayne; D Clive Williams; Mary J Meegan
Journal:  Pharmaceuticals (Basel)       Date:  2020-01-17

2.  C-H Amination via Electrophotocatalytic Ritter-type Reaction.

Authors:  Tao Shen; Tristan H Lambert
Journal:  J Am Chem Soc       Date:  2021-06-02       Impact factor: 16.383

3.  Manganese-catalysed benzylic C(sp3)-H amination for late-stage functionalization.

Authors:  Joseph R Clark; Kaibo Feng; Anasheh Sookezian; M Christina White
Journal:  Nat Chem       Date:  2018-04-30       Impact factor: 24.427

  3 in total

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