Literature DB >> 12620665

Synthesis and investigation of tuberculosis inhibition activities of some 1,2,3-triazole derivatives.

Kadir Dabak1, Ozkan Sezer, Ahmet Akar, Olcay Anaç.   

Abstract

In this study, alpha-diazo-beta-oxoaldehyde compounds were condensed with different amines to yield 4-acyl-1H-1,2,3-triazole derivatives. The 1,2,3-triazole compounds were investigated for their inhibition activities against tuberculosis.

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Year:  2003        PMID： 12620665     DOI： 10.1016/s0223-5234(02)01445-9

Source DB:  PubMed          Journal:  Eur J Med Chem        ISSN： 0223-5234            Impact factor:   6.514


  7 in total

1.  Targeting tuberculosis through a small focused library of 1,2,3-triazoles.

Authors:  Guillermo R Labadie; Agustina de la Iglesia; Héctor R Morbidoni
Journal:  Mol Divers       Date:  2011-06-02       Impact factor: 2.943

2.  α-Azido ketones. Part 7: synthesis of 1,4-disubstituted triazoles by the "click" reaction of various terminal acetylenes with phenacyl azides or α-azidobenzo(hetera)cyclanones.

Authors:  Krisztina Kónya; Szabolcs Fekete; Anita Abrahám; Tamás Patonay
Journal:  Mol Divers       Date:  2012-02-04       Impact factor: 2.943

3.  One-pot three-step synthesis of 1,2,3-triazoles by copper-catalyzed cycloaddition of azides with alkynes formed by a Sonogashira cross-coupling and desilylation.

Authors:  Frédéric Friscourt; Geert-Jan Boons
Journal:  Org Lett       Date:  2010-11-05       Impact factor: 6.005

4.  Antitubercular activity of 1,2,3-triazolyl fatty acid derivatives.

Authors:  Diego G Ghiano; Agustina de la Iglesia; Nina Liu; Peter J Tonge; Héctor R Morbidoni; Guillermo R Labadie
Journal:  Eur J Med Chem       Date:  2016-09-28       Impact factor: 6.514

5.  Synthesis of 1,2,3-triazole derivatives and in vitro antifungal evaluation on Candida strains.

Authors:  Reginaldo G Lima-Neto; Nery N M Cavalcante; Rajendra M Srivastava; Francisco J B Mendonça Junior; Almir G Wanderley; Rejane P Neves; Janaína V dos Anjos
Journal:  Molecules       Date:  2012-05-16       Impact factor: 4.411

6.  Synthesis of new 1,2,3-triazole derivatives of uracil and thymine with potential inhibitory activity against acidic corrosion of steels.

Authors:  Guillermo E Negrón-Silva; Rodrigo González-Olvera; Deyanira Angeles-Beltrán; Nidia Maldonado-Carmona; Araceli Espinoza-Vázquez; Manuel E Palomar-Pardavé; Mario A Romero-Romo; Rosa Santillan
Journal:  Molecules       Date:  2013-04-18       Impact factor: 4.411

7.  Design, Synthesis, and the Biological Evaluation of a New Series of Acyclic 1,2,3-Triazole Nucleosides.

Authors:  Iwona E Głowacka; Graciela Andrei; Dominique Schols; Robert Snoeck; Katarzyna Gawron
Journal:  Arch Pharm (Weinheim)       Date:  2017-08-01       Impact factor: 3.751
  7 in total

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