Literature DB >> 12491310

Click chemistry in situ: acetylcholinesterase as a reaction vessel for the selective assembly of a femtomolar inhibitor from an array of building blocks.

Warren G Lewis1, Luke G Green, Flavio Grynszpan, Zoran Radić, Paul R Carlier, Palmer Taylor, M G Finn, K Barry Sharpless.   

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Year:  2002        PMID： 12491310     DOI： 10.1002/1521-3773(20020315)41:6<1053::aid-anie1053>3.0.co;2-4

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


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  128 in total

1.  Structural insights into ligand interactions at the acetylcholinesterase peripheral anionic site.

Authors:  Yves Bourne; Palmer Taylor; Zoran Radić; Pascale Marchot
Journal:  EMBO J       Date:  2003-01-02       Impact factor: 11.598

Review 2.  Contemporary paradigms for cholinergic ligand design guided by biological structure.

Authors:  Palmer Taylor; Scott B Hansen; Todd T Talley; Ryan E Hibbs; Zoran Radić
Journal:  Bioorg Med Chem Lett       Date:  2004-04-19       Impact factor: 2.823

3.  N-activated β-lactams as versatile reagents for acyl carrier protein labeling.

Authors:  Gitanjeli Prasad; Jon W Amoroso; Lawrence S Borketey; Nathan A Schnarr
Journal:  Org Biomol Chem       Date:  2012-01-31       Impact factor: 3.876

4.  Hit clustering can improve virtual fragment screening: CDK2 and PARP1 case studies.

Authors:  Alexey A Zeifman; Victor S Stroylov; Fedor N Novikov; Oleg V Stroganov; Alexandra L Zakharenko; Svetlana N Khodyreva; Olga I Lavrik; Ghermes G Chilov
Journal:  J Mol Model       Date:  2011-11-09       Impact factor: 1.810

5.  A decade of chemical biology.

Authors:  Mirella Bucci; Catherine Goodman; Terry L Sheppard
Journal:  Nat Chem Biol       Date:  2010-12       Impact factor: 15.040

6.  A BODIPY-cyclooctyne for protein imaging in live cells.

Authors:  Kimberly E Beatty; Janek Szychowski; John D Fisk; David A Tirrell
Journal:  Chembiochem       Date:  2011-08-09       Impact factor: 3.164

7.  A Toxic RNA Templates the Synthesis of Its Own Fluorogenic Inhibitor by Using a Bio-orthogonal Tetrazine Ligation in Cells and Tissues.

Authors:  Alicia J Angelbello; Matthew D Disney
Journal:  ACS Chem Biol       Date:  2020-06-17       Impact factor: 5.100

8.  Fitness Factors for Bioorthogonal Chemical Probes.

Authors:  Yulin Tian; Qing Lin
Journal:  ACS Chem Biol       Date:  2019-12-05       Impact factor: 5.100

9.  Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor.

Authors:  Tomoyasu Hirose; Nobuo Maita; Hiroaki Gouda; Jun Koseki; Tsuyoshi Yamamoto; Akihiro Sugawara; Hirofumi Nakano; Shuichi Hirono; Kazuro Shiomi; Takeshi Watanabe; Hisaaki Taniguchi; K Barry Sharpless; Satoshi Omura; Toshiaki Sunazuka
Journal:  Proc Natl Acad Sci U S A       Date:  2013-09-16       Impact factor: 11.205

10.  Accurate MALDI-TOF/TOF sequencing of one-bead-one-compound peptide libraries with application to the identification of multiligand protein affinity agents using in situ click chemistry screening.

Authors:  Su Seong Lee; Jaehong Lim; Sylvia Tan; Junhoe Cha; Shi Yun Yeo; Heather D Agnew; James R Heath
Journal:  Anal Chem       Date:  2010-01-15       Impact factor: 6.986
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