Literature DB >> 12215937

[Dolasetron reduces pain on injection of propofol].

S N Piper1, K D Röhm, M Papsdorf, W H Maleck, P Mattinger, J Boldt.   

Abstract

OBJECTIVE: Pain on injection is a well known side-effect of propofol. The present study was designed to assess the efficacy of dolasetron, a 5-HT 3 -antagonist, in prophylaxis of pain on injection of propofol compared with lidocaine and placebo.
METHODS: Prospective, randomised, double-blinded study including 150 patients randomly assigned to one of three groups: Group A received 12.5 mg dolasetron, group B 40 mg lidocaine and group C saline 0.9 % as placebo. After occluding the venous drainage the test medication was given. The occlusion was released after 1 min and 2.0 mg/kg Propofol was administered over a period of 30 sec. The patients were asked whether they felt any pain during the administration. Pain on injection was judged by using a four-point scale.
RESULTS: Incidence of pain on injection as well as the severity of pain was significantly reduced by lidocaine (62 % pain free) compared with placebo (28 %). Severity, but not incidence of pain on injection was significantly reduced by dolasetron (50 %) compared with placebo. There was no significant difference between dolasetron and lidocaine.
CONCLUSION: Dolasetron and lidocaine were effective in preventing pain of injection secondary to propofol.

Entities:  

Year:  2002        PMID: 12215937     DOI: 10.1055/s-2002-33767

Source DB:  PubMed          Journal:  Anasthesiol Intensivmed Notfallmed Schmerzther        ISSN: 0939-2661            Impact factor:   0.698


  5 in total

Review 1.  The 5-HT3 receptor as a therapeutic target.

Authors:  Andrew J Thompson; Sarah C R Lummis
Journal:  Expert Opin Ther Targets       Date:  2007-04       Impact factor: 6.902

Review 2.  [Total intravenous anesthesia. On the way to standard practice in pediatrics].

Authors:  J M Strauss; J Giest
Journal:  Anaesthesist       Date:  2003-09       Impact factor: 1.041

3.  A comparative study of attenuation of propofol-induced pain by lignocaine, ondansetron, and ramosetron.

Authors:  Gangur Basappa Sumalatha; Ravichandra Ramesh Dodawad; Sandeep Pandarpurkar; Parashuram R Jajee
Journal:  Indian J Anaesth       Date:  2016-01

4.  Antimalarial drugs inhibit human 5-HT(3) and GABA(A) but not GABA(C) receptors.

Authors:  A J Thompson; S C R Lummis
Journal:  Br J Pharmacol       Date:  2008-03-03       Impact factor: 8.739

5.  Prevention of propofol injection pain: Comparison between lidocaine and ramosetron.

Authors:  Dipali Singh; Sathyanarayan Jagannath; Shio Priye; Chandrashekar Kadli; Durgaprasad Reddy
Journal:  J Anaesthesiol Clin Pharmacol       Date:  2014-04
  5 in total

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