Literature DB >> 12134506

A new binding mode of competitive antagonists to metabotropic glutamate receptors exemplified by the mGluR1-receptor antagonist AIDA (RS-aminoindan-1,5-dicarboxylic acid).

M S Belenikin1, I I Baskin, V A Palyulin, N S Zefirov.   

Abstract

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Year:  2002        PMID： 12134506     DOI： 10.1023/a:1016076028063

Source DB:  PubMed          Journal:  Dokl Biochem Biophys        ISSN： 1607-6729            Impact factor:   0.788


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  9 in total

1.  Q: a molecular dynamics program for free energy calculations and empirical valence bond simulations in biomolecular systems.

Authors:  J Marelius; K Kolmodin; I Feierberg; J Aqvist
Journal:  J Mol Graph Model       Date:  1998 Aug-Dec       Impact factor: 2.518

Review 2.  Metabotropic glutamate receptors: a structural view point.

Authors:  R Pellicciari; G Costantino; A Macchiarulo
Journal:  Pharm Acta Helv       Date:  2000-03

3.  Salt bridge stability in monomeric proteins.

Authors:  S Kumar; R Nussinov
Journal:  J Mol Biol       Date:  1999-11-12       Impact factor: 5.469

Review 4.  Pharmacological agents acting at subtypes of metabotropic glutamate receptors.

Authors:  D D Schoepp; D E Jane; J A Monn
Journal:  Neuropharmacology       Date:  1999-10       Impact factor: 5.250

Review 5.  Ligands for glutamate receptors: design and therapeutic prospects.

Authors:  H Bräuner-Osborne; J Egebjerg; E O Nielsen; U Madsen; P Krogsgaard-Larsen
Journal:  J Med Chem       Date:  2000-07-13       Impact factor: 7.446

6.  Modeling of amino-terminal domains of group I metabotropic glutamate receptors: structural motifs affecting ligand selectivity.

Authors:  G Costantino; A Macchiarulo; R Pellicciari
Journal:  J Med Chem       Date:  1999-12-30       Impact factor: 7.446

7.  Pharmacological characterization of 1-aminoindan-1,5-dicarboxylic acid, a potent mGluR1 antagonist.

Authors:  F Moroni; G Lombardi; C Thomsen; P Leonardi; S Attucci; F Peruginelli; S A Torregrossa; D E Pellegrini-Giampietro; R Luneia; R Pellicciari
Journal:  J Pharmacol Exp Ther       Date:  1997-05       Impact factor: 4.030

8.  Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor.

Authors:  N Kunishima; Y Shimada; Y Tsuji; T Sato; M Yamamoto; T Kumasaka; S Nakanishi; H Jingami; K Morikawa
Journal:  Nature       Date:  2000-10-26       Impact factor: 49.962

9.  Synthesis and preliminary evaluation of (S)-2-(4'-carboxycubyl)glycine, a new selective mGluR1 antagonist.

Authors:  R Pellicciari; G Costantino; E Giovagnoni; L Mattoli; I Brabet; J P Pin
Journal:  Bioorg Med Chem Lett       Date:  1998-06-16       Impact factor: 2.823
  9 in total

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