Literature DB >> 11959784

2-Chloro-N6-methyl-(N)-methanocarba-2'-deoxyadenosine-3',5'-bisphosphate is a selective high affinity P2Y1 receptor antagonist: commentary on Boyer et al.

Brian F King1.   

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Year:  2002        PMID： 11959784      PMCID： PMC1573331          DOI： 10.1038/sj.bjp.0704674

Source DB:  PubMed          Journal:  Br J Pharmacol        ISSN： 0007-1188            Impact factor:   8.739


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  9 in total

1.  Methanocarba modification of uracil and adenine nucleotides: high potency of Northern ring conformation at P2Y1, P2Y2, P2Y4, and P2Y11 but not P2Y6 receptors.

Authors:  Hak Sung Kim; R Gnana Ravi; Victor E Marquez; Savitri Maddileti; Anna-Karin Wihlborg; David Erlinge; Malin Malmsjö; José L Boyer; T Kendall Harden; Kenneth A Jacobson
Journal:  J Med Chem       Date:  2002-01-03       Impact factor: 7.446

2.  Identification of a novel human ADP receptor coupled to G(i).

Authors:  D Communi; N S Gonzalez; M Detheux; S Brézillon; V Lannoy; M Parmentier; J M Boeynaems
Journal:  J Biol Chem       Date:  2001-08-23       Impact factor: 5.157

3.  2-Chloro N(6)-methyl-(N)-methanocarba-2'-deoxyadenosine-3',5'-bisphosphate is a selective high affinity P2Y(1) receptor antagonist.

Authors:  José L Boyer; Mary Adams; R Gnana Ravi; Kenneth A Jacobson; T Kendall Harden
Journal:  Br J Pharmacol       Date:  2002-04       Impact factor: 8.739

4.  Identification of competitive antagonists of the P2Y1 receptor.

Authors:  J L Boyer; T Romero-Avila; J B Schachter; T K Harden
Journal:  Mol Pharmacol       Date:  1996-11       Impact factor: 4.436

5.  On the suitability of adenosine 3'-phosphate 5'-phosphosulphate as a selective P2Y receptor antagonist in intact tissues.

Authors:  R Bültmann; F Tuluc; K Starke
Journal:  Eur J Pharmacol       Date:  1998-06-19       Impact factor: 4.432

6.  Competitive and selective antagonism of P2Y1 receptors by N6-methyl 2'-deoxyadenosine 3',5'-bisphosphate.

Authors:  J L Boyer; A Mohanram; E Camaioni; K A Jacobson; T K Harden
Journal:  Br J Pharmacol       Date:  1998-05       Impact factor: 8.739

7.  Activity of Novel Adenine Nucleotide Derivatives as Agonists and Antagonists at Recombinant Rat P2X Receptors.

Authors:  Sean G Brown; Brian F King; Yong-Chul Kim; Soo Yeon Jang; Geoffrey Burnstock; Kenneth A Jacobson
Journal:  Drug Dev Res       Date:  2000-06-12       Impact factor: 4.360

8.  Cloning and functional expression of a brain G-protein-coupled ATP receptor.

Authors:  T E Webb; J Simon; B J Krishek; A N Bateson; T G Smart; B F King; G Burnstock; E A Barnard
Journal:  FEBS Lett       Date:  1993-06-14       Impact factor: 4.124

9.  Synthesis, biological activity, and molecular modeling of ribose-modified deoxyadenosine bisphosphate analogues as P2Y(1) receptor ligands.

Authors:  E Nandanan; S Y Jang; S Moro; H O Kim; M A Siddiqui; P Russ; V E Marquez; R Busson; P Herdewijn; T K Harden; J L Boyer; K A Jacobson
Journal:  J Med Chem       Date:  2000-03-09       Impact factor: 8.039
  9 in total
  1 in total

1.  P2Y(1) receptors mediate inhibitory neuromuscular transmission in the rat colon.

Authors:  Laura Grasa; Víctor Gil; Diana Gallego; Maria Teresa Martín; Marcel Jiménez
Journal:  Br J Pharmacol       Date:  2009-11       Impact factor: 8.739
  1 in total

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