Literature DB >> 11934243

Forecasting the oral absorption behavior of poorly soluble weak bases using solubility and dissolution studies in biorelevant media.

Edmund S Kostewicz1, Ulrich Brauns, Robert Becker, Jennifer B Dressman.   

Abstract

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Year:  2002        PMID： 11934243     DOI： 10.1023/a:1014407421366

Source DB:  PubMed          Journal:  Pharm Res        ISSN： 0724-8741            Impact factor:   4.200


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  9 in total

1.  Forecasting the in vivo performance of four low solubility drugs from their in vitro dissolution data.

Authors:  E Nicolaides; E Galia; C Efthymiopoulos; J B Dressman; C Reppas
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Review 2.  Dissolution testing as a prognostic tool for oral drug absorption: immediate release dosage forms.

Authors:  J B Dressman; G L Amidon; C Reppas; V P Shah
Journal:  Pharm Res       Date:  1998-01       Impact factor: 4.200

3.  The absolute and relative bioavailability of dipyridamole from different preparations and the in vitro-in vivo comparison.

Authors:  B Terhaag; F Donath; G Le Petit; K Feller
Journal:  Int J Clin Pharmacol Ther Toxicol       Date:  1986-06

4.  Upper gastrointestinal (GI) pH in young, healthy men and women.

Authors:  J B Dressman; R R Berardi; L C Dermentzoglou; T L Russell; S P Schmaltz; J L Barnett; K M Jarvenpaa
Journal:  Pharm Res       Date:  1990-07       Impact factor: 4.200

Review 5.  Influence of food on the bioavailability of drugs.

Authors:  A Melander
Journal:  Clin Pharmacokinet       Date:  1978 Sep-Oct       Impact factor: 6.447

6.  Solubilizing properties of bile salt solutions. I. Effect of temperature and bile salt concentration on solubilization of glutethimide, griseofulvin, and hexestrol.

Authors:  T R Bates; M Gibaldi; J L Kanig
Journal:  J Pharm Sci       Date:  1966-02       Impact factor: 3.534

7.  Intraluminal pH in the stomach, duodenum, and proximal jejunum in normal subjects and patients with exocrine pancreatic insufficiency.

Authors:  L Ovesen; F Bendtsen; U Tage-Jensen; N T Pedersen; B R Gram; S J Rune
Journal:  Gastroenterology       Date:  1986-04       Impact factor: 22.682

8.  Evaluation of various dissolution media for predicting in vivo performance of class I and II drugs.

Authors:  E Galia; E Nicolaides; D Hörter; R Löbenberg; C Reppas; J B Dressman
Journal:  Pharm Res       Date:  1998-05       Impact factor: 4.200

9.  pH-related changes in the absorption of dipyridamole in the elderly.

Authors:  T L Russell; R R Berardi; J L Barnett; T L O'Sullivan; J G Wagner; J B Dressman
Journal:  Pharm Res       Date:  1994-01       Impact factor: 4.200
  9 in total
  18 in total

1.  Administration of substances to laboratory animals: equipment considerations, vehicle selection, and solute preparation.

Authors:  Patricia V Turner; Cynthia Pekow; Mary Ann Vasbinder; Thea Brabb
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2.  Cocrystals Mitigate Negative Effects of High pH on Solubility and Dissolution of a Basic Drug.

Authors:  Yitian M Chen; Naír Rodríguez-Hornedo
Journal:  Cryst Growth Des       Date:  2018-02-14       Impact factor: 4.076

Review 3.  Biowaivers for oral immediate-release products: implications of linear pharmacokinetics.

Authors:  Fried Faassen; Herman Vromans
Journal:  Clin Pharmacokinet       Date:  2004       Impact factor: 6.447

4.  Predicting pharmacokinetic food effects using biorelevant solubility media and physiologically based modelling.

Authors:  Hannah M Jones; Neil Parrott; Gerd Ohlenbusch; Thierry Lavé
Journal:  Clin Pharmacokinet       Date:  2006       Impact factor: 6.447

Review 5.  Modeling kinetics of subcellular disposition of chemicals.

Authors:  Stefan Balaz
Journal:  Chem Rev       Date:  2009-05       Impact factor: 60.622

6.  Dissolution media simulating conditions in the proximal human gastrointestinal tract: an update.

Authors:  Ekarat Jantratid; Niels Janssen; Christos Reppas; Jennifer B Dressman
Journal:  Pharm Res       Date:  2008-04-11       Impact factor: 4.200

7.  pH-Induced precipitation behavior of weakly basic compounds: determination of extent and duration of supersaturation using potentiometric titration and correlation to solid state properties.

Authors:  Yi-Ling Hsieh; Grace A Ilevbare; Bernard Van Eerdenbrugh; Karl J Box; Manuel Vincente Sanchez-Felix; Lynne S Taylor
Journal:  Pharm Res       Date:  2012-05-12       Impact factor: 4.200

8.  In vivo bioequivalence and in vitro similarity factor (f2) for dissolution profile comparisons of extended release formulations: how and when do they match?

Authors:  John Z Duan; Kareen Riviere; Patrick Marroum
Journal:  Pharm Res       Date:  2011-02-02       Impact factor: 4.200

9.  Multivariate data analysis of factors affecting the in vitro dissolution rate and the apparent solubility for a model basic drug substance in aqueous media.

Authors:  Anita Maria Persson; Curt Pettersson; Josefin Rosén
Journal:  Pharm Res       Date:  2010-03-27       Impact factor: 4.200

10.  Colloid formation by drugs in simulated intestinal fluid.

Authors:  Allison K Doak; Holger Wille; Stanley B Prusiner; Brian K Shoichet
Journal:  J Med Chem       Date:  2010-05-27       Impact factor: 7.446
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