Literature DB >> 11921220

Crystallization-induced diastereoselection: asymmetric synthesis of substance P inhibitors.

Philip J Pye1, Kai Rossen, Steven A Weissman, Ashok Maliakal, Robert A Reamer, Richard Ball, Nancy N Tsou, R P Volante, Paul J Reider.   

Abstract

A novel three-component condensation followed by a crystallization-induced asymmetric transformation is used to build this key substance P inhibitor intermediate in a short synthetic sequence.

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Year:  2002        PMID： 11921220     DOI： 10.1002/1521-3765(20020315)8:6<1372::aid-chem1372>3.0.co;2-6

Source DB:  PubMed          Journal:  Chemistry        ISSN： 0947-6539            Impact factor:   5.236


  3 in total

1.  A novel route to synthesize libraries of quinoxalines via Petasis methodology in two synthetic operations.

Authors:  Muhammad Ayaz; Justin Dietrich; Christopher Hulme
Journal:  Tetrahedron Lett       Date:  2011-09-21       Impact factor: 2.415

2.  Doubly stereoconvergent crystallization enabled by asymmetric catalysis.

Authors:  Pedro de Jesús Cruz; William R Cassels; Chun-Hsing Chen; Jeffrey S Johnson
Journal:  Science       Date:  2022-06-09       Impact factor: 63.714

3.  Highly Efficient Synthesis of Optically Pure (S)-1-phenyl-1,2-ethanediol by a Self-Sufficient Whole Cell Biocatalyst.

Authors:  Xi Chen; Ting Mei; Yunfeng Cui; Qijia Chen; Xiangtao Liu; Jinhui Feng; Qiaqing Wu; Dunming Zhu
Journal:  ChemistryOpen       Date:  2015-04-30       Impact factor: 2.911
  3 in total

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