Literature DB >> 11594848

New ammonia equivalents for the Pd-catalyzed amination of aryl halides.

X Huang1, S L Buchwald.   

Abstract

[reaction: see text]. LiN(SiMe3)2, Ph3SiNH2, and LiNH2 can be be used as ammonia equivalents for the Pd-catalyzed coupling of aryl halides. Using these amine derivatives, simple anilines, including ortho-substituted ones, as well as di- and triarylamines can be readily prepared.

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Year:  2001        PMID： 11594848     DOI： 10.1021/ol0166808

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  14 in total

1.  Synthesis of Sterically Hindered Polychlorinated Biphenyl Derivatives.

Authors:  S N Joshi; S M Vyas; M W Duffel; S Parkin; H-J Lehmler
Journal:  Synthesis (Stuttg)       Date:  2011-01-01       Impact factor: 3.157

2.  Dialkylbiaryl Phosphines in Pd-Catalyzed Amination: A User's Guide.

Authors:  David S Surry; Stephen L Buchwald
Journal:  Chem Sci       Date:  2011       Impact factor: 9.825

3.  Discovery of a Novel Class of Imidazo[1,2-a]Pyridines with Potent PDGFR Activity and Oral Bioavailability.

Authors:  Erik J Hicken; Fred P Marmsater; Mark C Munson; Stephen T Schlachter; John E Robinson; Shelley Allen; Laurence E Burgess; Robert Kirk DeLisle; James P Rizzi; George T Topalov; Qian Zhao; Julie M Hicks; Nicholas C Kallan; Eugene Tarlton; Andrew Allen; Michele Callejo; April Cox; Sumeet Rana; Nathalie Klopfenstein; Richard Woessner; Joseph P Lyssikatos
Journal:  ACS Med Chem Lett       Date:  2013-11-12       Impact factor: 4.345

Review 4.  Catalytic organometallic reactions of ammonia.

Authors:  Jessica L Klinkenberg; John F Hartwig
Journal:  Angew Chem Int Ed Engl       Date:  2011-01-03       Impact factor: 15.336

5.  Design, synthesis, and biological evaluation of 3,4-dihydroquinolin-2(1H)-one and 1,2,3,4-tetrahydroquinoline-based selective human neuronal nitric oxide synthase (nNOS) inhibitors.

Authors:  Jailall Ramnauth; Joanne Speed; Shawn P Maddaford; Peter Dove; Subhash C Annedi; Paul Renton; Suman Rakhit; John Andrews; Sarah Silverman; Gabriela Mladenova; Salvatore Zinghini; Sheela Nair; Concettina Catalano; David K H Lee; Milena De Felice; Frank Porreca
Journal:  J Med Chem       Date:  2011-07-08       Impact factor: 7.446

6.  A novel, unusually efficacious duocarmycin carbamate prodrug that releases no residual byproduct.

Authors:  Amanda L Wolfe; Katharine K Duncan; Nikhil K Parelkar; Scott J Weir; George A Vielhauer; Dale L Boger
Journal:  J Med Chem       Date:  2012-06-12       Impact factor: 7.446

7.  A concise silylamine approach to 2-amino-3-hydroxy-indoles with potent in vivo antimalaria activity.

Authors:  Sameer Urgaonkar; Joseph F Cortese; Robert H Barker; Mandy Cromwell; Adelfa E Serrano; Dyann F Wirth; Jon Clardy; Ralph Mazitschek
Journal:  Org Lett       Date:  2010-09-17       Impact factor: 6.005

8.  Installation of protected ammonia equivalents onto aromatic & heteroaromatic rings in water enabled by micellar catalysis.

Authors:  Nicholas A Isley; Sebastian Dobarco; Bruce H Lipshutz
Journal:  Green Chem       Date:  2014-01-02       Impact factor: 10.182

9.  Mild and highly selective palladium-catalyzed monoarylation of ammonia enabled by the use of bulky biarylphosphine ligands and palladacycle precatalysts.

Authors:  Chi Wai Cheung; David S Surry; Stephen L Buchwald
Journal:  Org Lett       Date:  2013-07-01       Impact factor: 6.005

Review 10.  Applications of Palladium-Catalyzed C-N Cross-Coupling Reactions.

Authors:  Paula Ruiz-Castillo; Stephen L Buchwald
Journal:  Chem Rev       Date:  2016-09-30       Impact factor: 60.622
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