Literature DB >> 11495577

The first potent and selective inhibitors of the glycine transporter type 2.

W L Caulfield1, I T Collie, R S Dickins, O Epemolu, R McGuire, D R Hill, G McVey, J R Morphy, Z Rankovic, H Sundaram.   

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Year:  2001        PMID： 11495577     DOI： 10.1021/jm0011272

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  20 in total

Review 1.  The solute carrier 6 family of transporters.

Authors:  Stefan Bröer; Ulrik Gether
Journal:  Br J Pharmacol       Date:  2012-09       Impact factor: 8.739

2.  The transporters GlyT2 and VIAAT cooperate to determine the vesicular glycinergic phenotype.

Authors:  Karin R Aubrey; Francesco M Rossi; Raquel Ruivo; Silvia Alboni; Gian Carlo Bellenchi; Anne Le Goff; Bruno Gasnier; Stéphane Supplisson
Journal:  J Neurosci       Date:  2007-06-06       Impact factor: 6.167

3.  Activation of a glycine transporter on spinal cord neurons causes enhanced glutamate release in a mouse model of amyotrophic lateral sclerosis.

Authors:  Luca Raiteri; Egle Paolucci; Simona Prisco; Maurizio Raiteri; Giambattista Bonanno
Journal:  Br J Pharmacol       Date:  2003-03       Impact factor: 8.739

4.  P2Y purinergic regulation of the glycine neurotransmitter transporters.

Authors:  Esperanza Jiménez; Francisco Zafra; Raquel Pérez-Sen; Esmerilda G Delicado; Maria Teresa Miras-Portugal; Carmen Aragón; Beatriz López-Corcuera
Journal:  J Biol Chem       Date:  2011-01-18       Impact factor: 5.157

5.  Bergmann glial GlyT1 mediates glycine uptake and release in mouse cerebellar slices.

Authors:  Hao Huang; Latifa Barakat; Doris Wang; Angélique Bordey
Journal:  J Physiol       Date:  2004-08-26       Impact factor: 5.182

6.  Reversible inhibition of the glycine transporter GlyT2 circumvents acute toxicity while preserving efficacy in the treatment of pain.

Authors:  A Mingorance-Le Meur; P Ghisdal; B Mullier; P De Ron; P Downey; C Van Der Perren; V Declercq; S Cornelis; M Famelart; J Van Asperen; E Jnoff; J P Courade
Journal:  Br J Pharmacol       Date:  2013-11       Impact factor: 8.739

7.  Role of glial and neuronal glycine transporters in the control of glycinergic and glutamatergic synaptic transmission in lamina X of the rat spinal cord.

Authors:  Amyaouch Bradaïa; Rémy Schlichter; Jérôme Trouslard
Journal:  J Physiol       Date:  2004-07-02       Impact factor: 5.182

8.  GABAA and glycine receptor-mediated transmission in rat lamina II neurones: relevance to the analgesic actions of neuroactive steroids.

Authors:  Elizabeth A Mitchell; Luc J Gentet; John Dempster; Delia Belelli
Journal:  J Physiol       Date:  2007-07-26       Impact factor: 5.182

Review 9.  Heteromeric Solute Carriers: Function, Structure, Pathology and Pharmacology.

Authors:  Stephen J Fairweather; Nishank Shah; Stefan Brӧer
Journal:  Adv Exp Med Biol       Date:  2021       Impact factor: 2.622

10.  Development of an N-Acyl Amino Acid That Selectively Inhibits the Glycine Transporter 2 To Produce Analgesia in a Rat Model of Chronic Pain.

Authors:  Shannon N Mostyn; Tristan Rawling; Sarasa Mohammadi; Susan Shimmon; Zachary J Frangos; Subhodeep Sarker; Arsalan Yousuf; Irina Vetter; Renae M Ryan; Macdonald J Christie; Robert J Vandenberg
Journal:  J Med Chem       Date:  2019-02-20       Impact factor: 7.446
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