Literature DB >> 11460825

Insurmountable AT(1) receptor antagonism: the need for different antagonist binding states of the receptor.

G Vauquelin, F Fierens, I Verheijen, P Vanderheyden.   

Abstract

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Year:  2001        PMID： 11460825     DOI： 10.1016/s0165-6147(00)01739-9

Source DB:  PubMed          Journal:  Trends Pharmacol Sci        ISSN： 0165-6147            Impact factor:   14.819


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  7 in total

Review 1.  Long-lasting target binding and rebinding as mechanisms to prolong in vivo drug action.

Authors:  Georges Vauquelin; Steven J Charlton
Journal:  Br J Pharmacol       Date:  2010-10       Impact factor: 8.739

2.  Estimation of the dissociation rate of unlabelled ligand-receptor complexes by a 'two-step' competition binding approach.

Authors:  A Packeu; M Wennerberg; A Balendran; G Vauquelin
Journal:  Br J Pharmacol       Date:  2010-11       Impact factor: 8.739

3.  Conformational switch of angiotensin II type 1 receptor underlying mechanical stress-induced activation.

Authors:  Noritaka Yasuda; Shin-ichiro Miura; Hiroshi Akazawa; Toshimasa Tanaka; Yingjie Qin; Yoshihiro Kiya; Satoshi Imaizumi; Masahiro Fujino; Kaoru Ito; Yunzeng Zou; Shigetomo Fukuhara; Satoshi Kunimoto; Koichi Fukuzaki; Toshiaki Sato; Junbo Ge; Naoki Mochizuki; Haruaki Nakaya; Keijiro Saku; Issei Komuro
Journal:  EMBO Rep       Date:  2008-01-18       Impact factor: 8.807

4.  A study of the molecular mechanism of binding kinetics and long residence times of human CCR5 receptor small molecule allosteric ligands.

Authors:  David C Swinney; Paul Beavis; Kai-Ting Chuang; Yue Zheng; Ina Lee; Peter Gee; Jerome Deval; David M Rotstein; Marianna Dioszegi; Palani Ravendran; Jun Zhang; Surya Sankuratri; Rama Kondru; Georges Vauquelin
Journal:  Br J Pharmacol       Date:  2014-07       Impact factor: 8.739

5.  Molecular characterisation of the interactions between olmesartan and telmisartan and the human angiotensin II AT1 receptor.

Authors:  M T Le; M K Pugsley; G Vauquelin; I Van Liefde
Journal:  Br J Pharmacol       Date:  2007-06-18       Impact factor: 8.739

6.  Characterization of a fluorescent conjugate of the rabbit angiotensin AT(1) receptor.

Authors:  Jean-Philippe Fortin; Johanne Bouthillier; Luc Bastien; Dimcho R Bachvarov; François Marceau
Journal:  Br J Pharmacol       Date:  2003-04       Impact factor: 8.739

Review 7.  The renin-angiotensin system in the brain: possible therapeutic implications for AT(1)-receptor blockers.

Authors:  J Culman; A Blume; P Gohlke; T Unger
Journal:  J Hum Hypertens       Date:  2002-08       Impact factor: 3.012
  7 in total

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