Literature DB >> 11440576

First total synthesis of martinellic acid, a naturally occurring bradykinin receptor antagonist.

D Ma1, C Xia, J Jiang, J Zhang.   

Abstract

[reaction: see text] The first total synthesis of martinellic acid, a naturally occurring bradykinin receptor antagonist, via a CuI-catalyzed coupling reaction of beta-amino ester 6 with 1,4-diiodobenzene and a guanylation reaction of secondary amine 3 under mild conditions as key steps, is described.

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Year:  2001        PMID： 11440576     DOI： 10.1021/ol016043h

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  8 in total

1.  Synthesis, molecular modeling and biological evaluation of aza-flavanones as α-glucosidase inhibitors.

Authors:  Sivaprasad Kasturi; Sujatha Surarapu; Chandra Chary Bathoju; Srinivas Uppalanchi; Shubham Dwivedi; Yogeeswari Perumal; Dilep Kumar Sigalapalli; Bathini Nagendra Babu; Krishna S Ethiraj; Jaya Shree Anireddy
Journal:  Medchemcomm       Date:  2017-06-14       Impact factor: 3.597

2.  Synthesis of phidianidines A and B.

Authors:  Hong-Yu Lin; Barry B Snider
Journal:  J Org Chem       Date:  2012-05-01       Impact factor: 4.354

3.  Synthesis of (+)- and (-)-monanchorin.

Authors:  Min Yu; Barry B Snider
Journal:  Org Lett       Date:  2009-02-19       Impact factor: 6.005

4.  Palladium- and copper-mediated N-aryl bond formation reactions for the synthesis of biological active compounds.

Authors:  Carolin Fischer; Burkhard Koenig
Journal:  Beilstein J Org Chem       Date:  2011-01-14       Impact factor: 2.883

5.  Synthesis, characterisation and reactivity of copper(I) amide complexes and studies on their role in the modified Ullmann amination reaction.

Authors:  Simon Sung; D Christopher Braddock; Alan Armstrong; Colin Brennan; David Sale; Andrew J P White; Robert P Davies
Journal:  Chemistry       Date:  2015-03-18       Impact factor: 5.236

6.  Kinetic resolution of racemic 2-substituted 1,2-dihydroquinolines via asymmetric Cu-catalyzed borylation.

Authors:  Duanyang Kong; Suna Han; Rui Wang; Meina Li; Guofu Zi; Guohua Hou
Journal:  Chem Sci       Date:  2017-04-19       Impact factor: 9.825

7.  Cu(I)-Catalyzed Alkynylation of Quinolones.

Authors:  Aitor Maestro; Sebastien Lemaire; Syuzanna R Harutyunyan
Journal:  Org Lett       Date:  2022-01-31       Impact factor: 6.005

8.  Copper(II)-Catalyzed (3+2) Cycloaddition of 2H-Azirines to Six-Membered Cyclic Enols as a Route to Pyrrolo[3,2-c]quinolone, Chromeno[3,4-b]pyrrole, and Naphtho[1,8-ef]indole Scaffolds.

Authors:  Pavel A Sakharov; Nikolai V Rostovskii; Alexander F Khlebnikov; Mikhail S Novikov
Journal:  Molecules       Date:  2022-09-02       Impact factor: 4.927
  8 in total

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