Literature DB >> 11310610

Synthesis of indomethacin analogues for evaluation as modulators of MRP activity.

A R Maguire1, S J Plunkett, S Papot, M Clynes, R O'Connor, S Touhey.   

Abstract

Synthesis of a range of indomethacin analogues, required for investigation in combination toxicity assays, bearing both N-benzyl and N-benzoyl groups, is described.

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Year:  2001        PMID： 11310610     DOI： 10.1016/s0968-0896(00)00292-3

Source DB:  PubMed          Journal:  Bioorg Med Chem        ISSN： 0968-0896            Impact factor:   3.641


  8 in total

1.  Increase in multidrug transport activity is associated with oocyte maturation in sea stars.

Authors:  Troy A Roepke; Amro M Hamdoun; Gary N Cherr
Journal:  Dev Growth Differ       Date:  2006-12       Impact factor: 2.053

2.  Ortho-carbaborane derivatives of indomethacin as cyclooxygenase (COX)-2 selective inhibitors.

Authors:  Matthias Scholz; Anna L Blobaum; Lawrence J Marnett; Evamarie Hey-Hawkins
Journal:  Bioorg Med Chem       Date:  2012-06-05       Impact factor: 3.641

3.  Catalytic ester-amide exchange using group (IV) metal alkoxide-activator complexes.

Authors:  Chong Han; Jonathan P Lee; Emil Lobkovsky; John A Porco
Journal:  J Am Chem Soc       Date:  2005-07-20       Impact factor: 15.419

4.  Straightforward protocol for the efficient synthesis of varied N(1)-acylated (aza)indole 2-/3-alkanoic acids and esters: optimization and scale-up.

Authors:  Andy J Liedtke; Kwangho Kim; Donald F Stec; Gary A Sulikowski; Lawrence J Marnett
Journal:  Tetrahedron       Date:  2012-12-02       Impact factor: 2.457

5.  Involvement of P-glycoprotein and multidrug resistance associated protein 1 on the transepithelial transport of a mercaptoacetamide-based histone-deacetylase inhibitor in Caco-2 cells.

Authors:  Zacharoula Konsoula; Mira Jung
Journal:  Biol Pharm Bull       Date:  2009-01       Impact factor: 2.233

6.  Inhibition of acetylcholinesterase by chromophore-linked fluorophosphonates.

Authors:  Lilu Guo; Alirica I Suarez; Michael R Braden; John M Gerdes; Charles M Thompson
Journal:  Bioorg Med Chem Lett       Date:  2009-12-04       Impact factor: 2.823

7.  Synthesis and biological evaluation of novel quinoline analogs of ketoprofen as multidrug resistance protein 2 (MRP2) inhibitors.

Authors:  Fatemeh Mosaffa; Farzin Hadizadeh; Faezeh Fathi; Zahra Eslami Nasab; Tahereh Pourzahed; Sayyed Mohammad Aboutorabzade; Razieh Ghodsi
Journal:  Iran J Basic Med Sci       Date:  2021-06       Impact factor: 2.699

8.  2-[5-Bromo-1-(3-chloro-benz-yl)-2-methyl-1H-indol-3-yl]acetic acid.

Authors:  Mahmoud Elkady; Peter R W E F Keck; Dieter Schollmeyer; Stefan Laufer
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-11-24
  8 in total

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