Literature DB >> 11152032

Plasma concentrations and pharmacokinetics of bupivacaine with and without adrenaline following caudal anaesthesia in infants.

T G Hansen1, N S Morton, P M Cullen, D G Watson.   

Abstract

BACKGROUND: The aim of this study was to determine whether the use of adrenaline 1/400000 added to 0.25% bupivacaine significantly delays the systemic absorption of the drug from the caudal epidural space in young infants.
METHODS: Fifteen infants less than 5 months of age undergoing minor lower abdominal procedures under a standardised general anaesthetic were randomised to receive a caudal block with either 0.25% plain bupivacaine 2.5 mg/kg (n=7) or bupivacaine 0.25% with 1/400000 adrenaline (n=8). Blood samples were drawn at 30, 60, 90, 180, 240 and 360 min according to the infant's weight and analysed for total and free bupivacaine concentrations using a gas chromatography-mass spectrometry (GC-MS) technique.
RESULTS: The total C(MAX) and T(MAX) were comparable in both groups. The total bupivacaine concentration at t=360 min was significantly higher in the "adrenaline" group compared to the "plain" group, i.e. a median (range) 742 ng/ml (372-1423 ng/ml) vs. 400.5 ng/ml (114-446 ng/ml), P=0.0080. The median "apparent" terminal half-life (t1/2) was significantly longer in the "adrenaline" group (363 min; range 238-537 min) compared to the "plain" group (n=6) (165 min; range 104-264 min), P=0.0087. The free bupivacaine concentrations (n=3 in both groups) ranged between 13 ng/ml and 52 ng/ml, corresponding to a percentage of free bupivacaine between 1.3% and 6.7%.
CONCLUSION: The addition of 1/400.000 adrenaline prolongs the systemic absorption of caudally administered bupivacaine in infants less than 5 months of age.

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Year:  2001        PMID: 11152032     DOI: 10.1034/j.1399-6576.2001.450107.x

Source DB:  PubMed          Journal:  Acta Anaesthesiol Scand        ISSN: 0001-5172            Impact factor:   2.105


  3 in total

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Authors:  Monika Daubländer; Peer W Kämmerer; Brita Willershausen; Michael Leckel; Hans-Christoph Lauer; Siegmar Buff; Benita Rösl
Journal:  Clin Oral Investig       Date:  2011-08-23       Impact factor: 3.573

Review 2.  Pharmacokinetics of local anaesthetics in infants and children.

Authors:  Jean-Xavier Mazoit; Bernard J Dalens
Journal:  Clin Pharmacokinet       Date:  2004       Impact factor: 6.447

3.  Epinephrine-reduced articaine solution (1:400,000) in paediatric dentistry: a multicentre non-interventional clinical trial.

Authors:  P W Kämmerer; N Krämer; J Esch; H Pfau; U Uhlemann; L Piehlmeier; M Daubländer
Journal:  Eur Arch Paediatr Dent       Date:  2013-04-05
  3 in total

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