Literature DB >> 9926287

Kinin receptors.

F Marceau1, D R Bachvarov.   

Abstract

Rapid developments are expected in the molecular pharmacology of both B1, and B2 types of kinin receptors, since the underlying genetic structures are now known and widely studied. The consequences of kinin receptor duality and physiopathological regulation have not yet been fully appreciated. Medicinal chemistry is also an active front of research in kinin pharmacology, as more effective drugs targeted at kinin receptors are regularly reported. Various complementary molecular approaches (the receptor binding, cloning, immunoreacting, mutagenesis, inactivation, the study of regulation, allelic polymorphisms, and so forth) are expanding our knowledge of the role of kinins in allergy, inflammation, and singularly, renal medicine.

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Year:  1998        PMID: 9926287     DOI: 10.1007/BF02737658

Source DB:  PubMed          Journal:  Clin Rev Allergy Immunol        ISSN: 1080-0549            Impact factor:   8.667


  79 in total

1.  Molecular cloning, functional expression and pharmacological characterization of a human bradykinin B2 receptor gene.

Authors:  D Eggerickx; E Raspe; D Bertrand; G Vassart; M Parmentier
Journal:  Biochem Biophys Res Commun       Date:  1992-09-30       Impact factor: 3.575

2.  An enzyme in human blood plasma that inactivates bradykinin and kallidins.

Authors:  E G ERDOS; E M SLOANE
Journal:  Biochem Pharmacol       Date:  1962-07       Impact factor: 5.858

3.  Mechanisms of endothelium-dependent vascular smooth muscle relaxation elicited by bradykinin and VIP.

Authors:  L J Ignarro; R E Byrns; G M Buga; K S Wood
Journal:  Am J Physiol       Date:  1987-11

4.  Bradykinin as a pain mediator: receptors are localized to sensory neurons, and antagonists have analgesic actions.

Authors:  L R Steranka; D C Manning; C J DeHaas; J W Ferkany; S A Borosky; J R Connor; R J Vavrek; J M Stewart; S H Snyder
Journal:  Proc Natl Acad Sci U S A       Date:  1988-05       Impact factor: 11.205

5.  Expression cloning of a rat B2 bradykinin receptor.

Authors:  A E McEachern; E R Shelton; S Bhakta; R Obernolte; C Bach; P Zuppan; J Fujisaki; R W Aldrich; K Jarnagin
Journal:  Proc Natl Acad Sci U S A       Date:  1991-09-01       Impact factor: 11.205

6.  [3H]Bradykinin receptor binding in mammalian tissue membranes.

Authors:  R B Innis; D C Manning; J M Stewart; S H Snyder
Journal:  Proc Natl Acad Sci U S A       Date:  1981-04       Impact factor: 11.205

7.  Contractions induced by angiotensin I, angiotensin II and bradykinin in isolated smooth muscle from the human detrusor.

Authors:  K E Andersson; H Hedlund; M Stahl
Journal:  Acta Physiol Scand       Date:  1992-07

8.  Competitive antagonists of bradykinin.

Authors:  R J Vavrek; J M Stewart
Journal:  Peptides       Date:  1985 Mar-Apr       Impact factor: 3.750

9.  Characterization of solubilized bradykinin B2 receptors from smooth muscle and mucosa of guinea pig ileum.

Authors:  R W Ransom; G S Young; K Schneck; C B Goodman
Journal:  Biochem Pharmacol       Date:  1992-04-15       Impact factor: 5.858

10.  Cloning and pharmacological characterization of a human bradykinin (BK-2) receptor.

Authors:  J F Hess; J A Borkowski; G S Young; C D Strader; R W Ransom
Journal:  Biochem Biophys Res Commun       Date:  1992-04-15       Impact factor: 3.575

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  34 in total

1.  Attenuation of persistent experimental pancreatitis pain by a bradykinin b2 receptor antagonist.

Authors:  Qingmin Chen; Louis P Vera-Portocarrero; Michael H Ossipov; Marina Vardanyan; Josephine Lai; Frank Porreca
Journal:  Pancreas       Date:  2010-11       Impact factor: 3.327

2.  Cytokines and neutrophils as important mediators of platelet-activating factor-induced kinin B1 receptor expression.

Authors:  Elizabeth S Fernandes; Giselle F Passos; Maria M Campos; Glória E P de Souza; Juliana F Fittipaldi; Jorge L Pesquero; Mauro M Teixeira; João B Calixto
Journal:  Br J Pharmacol       Date:  2005-09       Impact factor: 8.739

3.  Molecular and pharmacological evidence for modulation of kinin B(1) receptor expression by endogenous glucocorticoids hormones in rats.

Authors:  D A Cabrini; M M Campos; K S Tratsk; V F Merino; J A Silva ; G E Souza; M C Avellar; J B Pesquero; J B Calixto
Journal:  Br J Pharmacol       Date:  2001-01       Impact factor: 8.739

4.  Mechanisms underlying the modulatory action of platelet activating factor (PAF) on the upregulation of kinin B1 receptors in the rat paw.

Authors:  Elizabeth S Fernandes; Giselle F Passos; Maria M Campos; José G V C Araújo; Jorge L Pesquero; Maria C Avelllar; Mauro M Teixeira; João B Calixto
Journal:  Br J Pharmacol       Date:  2003-07       Impact factor: 8.739

5.  Wortmannin alters the intracellular trafficking of the bradykinin B2 receptor: role of phosphoinositide 3-kinase and Rab5.

Authors:  Steeve Houle; François Marceau
Journal:  Biochem J       Date:  2003-10-01       Impact factor: 3.857

Review 6.  Perspectives on the Trypanosoma cruzi-host cell receptor interactions.

Authors:  Fernando Villalta; Julio Scharfstein; Anthony W Ashton; Kevin M Tyler; Fangxia Guan; Shankar Mukherjee; Maria F Lima; Sandra Alvarez; Louis M Weiss; Huan Huang; Fabiana S Machado; Herbert B Tanowitz
Journal:  Parasitol Res       Date:  2009-03-13       Impact factor: 2.289

7.  Implication of the bradykinin receptors in antigen-induced pulmonary inflammation in mice.

Authors:  Jadranka Eric; Bichoy H Gabra; Pierre Sirois
Journal:  Br J Pharmacol       Date:  2003-04       Impact factor: 8.739

8.  Synergistic interaction between enalapril, L-arginine and tetrahydrobiopterin in smooth muscle cell apoptosis and aortic remodeling induction in SHR.

Authors:  Shant Der Sarkissian; Eve-Lyne Marchand; David Duguay; Denis deBlois
Journal:  Br J Pharmacol       Date:  2004-06-14       Impact factor: 8.739

9.  Cellular localization of kinin B1 receptor in the spinal cord of streptozotocin-diabetic rats with a fluorescent [Nalpha-Bodipy]-des-Arg9-bradykinin.

Authors:  Sébastien Talbot; Patrick Théberge-Turmel; Dalinda Liazoghli; Jacques Sénécal; Pierrette Gaudreau; Réjean Couture
Journal:  J Neuroinflammation       Date:  2009-03-26       Impact factor: 8.322

10.  Immunohistochemical localization of the bradykinin B1 and B2 receptors in human nasal mucosa.

Authors:  Hideaki Shirasaki; Etsuko Kanaizumi; Tetsuo Himi
Journal:  Mediators Inflamm       Date:  2009-04-23       Impact factor: 4.711

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