Literature DB >> 9925725

Discovery of a potent, orally active, nonsteroidal androgen receptor agonist: 4-ethyl-1,2,3,4-tetrahydro-6- (trifluoromethyl)-8-pyridono[5,6-g]- quinoline (LG121071).

L G Hamann1, N S Mani, R L Davis, X N Wang, K B Marschke, T K Jones.   

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Year:  1999        PMID： 9925725     DOI： 10.1021/jm9806648

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  10 in total

Review 1.  Chemistry and structural biology of androgen receptor.

Authors:  Wenqing Gao; Casey E Bohl; James T Dalton
Journal:  Chem Rev       Date:  2005-09       Impact factor: 60.622

2.  Photocytotoxicity of the fluorescent nonsteroidal androgen receptor ligand TDPQ.

Authors:  Piotr J Bilski; Boris Risek; Colin F Chignell; William T Schrader
Journal:  Photochem Photobiol       Date:  2009-05-28       Impact factor: 3.421

Review 3.  Pharmacokinetics and pharmacodynamics of nonsteroidal androgen receptor ligands.

Authors:  Wenqing Gao; Juhyun Kim; James T Dalton
Journal:  Pharm Res       Date:  2006-08       Impact factor: 4.200

Review 4.  Selective androgen receptor modulators as function promoting therapies.

Authors:  Shalender Bhasin; Ravi Jasuja
Journal:  Curr Opin Clin Nutr Metab Care       Date:  2009-05       Impact factor: 4.294

5.  Design, synthesis, and biological characterization of metabolically stable selective androgen receptor modulators.

Authors:  Craig A Marhefka; Wenqing Gao; Kiwon Chung; Juhyun Kim; Yali He; Donghua Yin; Casey Bohl; James T Dalton; Duane D Miller
Journal:  J Med Chem       Date:  2004-02-12       Impact factor: 7.446

Review 6.  Medicinal Use of Testosterone and Related Steroids Revisited.

Authors:  Jan Tauchen; Michal Jurášek; Lukáš Huml; Silvie Rimpelová
Journal:  Molecules       Date:  2021-02-15       Impact factor: 4.411

7.  Therapeutic androgen receptor ligands.

Authors:  George F Allan; Zhihua Sui
Journal:  Nucl Recept Signal       Date:  2003-09-27

Review 8.  Selective androgen receptor modulators in preclinical and clinical development.

Authors:  Ramesh Narayanan; Michael L Mohler; Casey E Bohl; Duane D Miller; James T Dalton
Journal:  Nucl Recept Signal       Date:  2008-11-26

Review 9.  Is There Room for SERMs or SARMs as Alternative Therapies for Adult Male Hypogonadism?

Authors:  Vito A Giagulli; Andrea Silvestrini; Carmine Bruno; Vincenzo Triggiani; Alvaro Mordente; Antonio Mancini
Journal:  Int J Endocrinol       Date:  2020-01-21       Impact factor: 3.257

10.  Nucleophilic Dearomatization of N-Heteroaromatics Enabled by Lewis Acids and Copper Catalysis.

Authors:  Xingchen Yan; Luo Ge; Marta Castiñeira Reis; Syuzanna R Harutyunyan
Journal:  J Am Chem Soc       Date:  2020-11-10       Impact factor: 15.419
  10 in total

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