Literature DB >> 9548811

4-Amino-2-[4-[1-(benzyloxycarbonyl)-2(S)- [[(1,1-dimethylethyl)amino]carbonyl]-piperazinyl]-6, 7-dimethoxyquinazoline (L-765,314): a potent and selective alpha1b adrenergic receptor antagonist.

M A Patane1, A L Scott, T P Broten, R S Chang, R W Ransom, J DiSalvo, C Forray, M G Bock.   

Abstract

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Year:  1998        PMID： 9548811     DOI： 10.1021/jm980053f

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  8 in total

1.  The role of several alpha(1)- and alpha(2)-adrenoceptor subtypes mediating vasoconstriction in the canine external carotid circulation.

Authors:  E W Willems; L F Valdivia; P R Saxena; C M Villalón
Journal:  Br J Pharmacol       Date:  2001-03       Impact factor: 8.739

2.  Interaction between alpha(1)- and alpha(2)-adrenoreceptors contributes to enhanced constrictor effects of norepinephrine in mesenteric veins compared to arteries.

Authors:  Alexandra Sporkova; Alex Perez-Rivera; James J Galligan
Journal:  Eur J Pharmacol       Date:  2010-06-21       Impact factor: 4.432

3.  Pharmacologically distinct phenotypes of α1B -adrenoceptors: variation in binding and functional affinities for antagonists.

Authors:  Hatsumi Yoshiki; Junsuke Uwada; Abu Syed Md Anisuzzaman; Hidenori Umada; Ryoji Hayashi; Mie Kainoh; Takayoshi Masuoka; Matomo Nishio; Ikunobu Muramatsu
Journal:  Br J Pharmacol       Date:  2014-09-05       Impact factor: 8.739

4.  Chiral analogues of (+)-cyclazosin as potent α1B-adrenoceptor selective antagonist.

Authors:  Gianni Sagratini; Michela Buccioni; Gabriella Marucci; Elena Poggesi; Matthew Skorski; Stefano Costanzi; Dario Giardinà
Journal:  Bioorg Med Chem       Date:  2018-05-17       Impact factor: 3.641

5.  alpha-Adrenoceptor-mediated depletion of phosphatidylinositol 4, 5-bisphosphate inhibits activation of volume-regulated anion channels in mouse ventricular myocytes.

Authors:  K Ichishima; S Yamamoto; T Iwamoto; T Ehara
Journal:  Br J Pharmacol       Date:  2010-09       Impact factor: 8.739

6.  Smooth muscle alpha1D-adrenoceptors mediate phenylephrine-induced vasoconstriction and increases in endothelial cell Ca2+ in hamster cremaster arterioles.

Authors:  W F Jackson; E M Boerman; E J Lange; S S Lundback; K D Cohen
Journal:  Br J Pharmacol       Date:  2008-07-07       Impact factor: 8.739

7.  Enhancement of apomorphine-induced penile erection in the rat by a selective alpha(1D)-adrenoceptor antagonist.

Authors:  Hiroya Mizusawa; Petter Hedlund; Johan Sjunnesson; Jorge D Brioni; James P Sullivan; Karl-Erik Andersson
Journal:  Br J Pharmacol       Date:  2002-07       Impact factor: 8.739

8.  The role of α1- and α2-adrenoceptor subtypes in the vasopressor responses induced by dihydroergotamine in ritanserin-pretreated pithed rats.

Authors:  Eduardo Rivera-Mancilla; Victor H Avilés-Rosas; Guadalupe Manrique-Maldonado; Alain H Altamirano-Espinoza; Belinda Villanueva-Castillo; Antoinette MaassenVanDenBrink; Carlos M Villalón
Journal:  J Headache Pain       Date:  2017-10-11       Impact factor: 7.277
  8 in total

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