Literature DB >> 9345343

Irinotecan hydrochloride (CPT-11) resistance identified by K-ras mutation in patients with progressive colon cancer after treatment with 5-fluorouracil (5-FU).

J Nemunaitis1, J Cox, W Meyer, A Courtney, G Mues.   

Abstract

OBJECTIVE: To determine the prognostic role of a K-ras mutation in tumor tissue of patients with refractory colon cancer who received irinotecan hydrochloride (CPT-11).
METHODS: DNA was extracted from paraffin-stored tumor tissue of 35 patients with progressive colon cancer failing treatment with 5-fluorouracil who subsequently received CPT-11 (100 mg/m2 i.v. per week x 4 weeks with 2 weeks off per course). The first exon of the K-ras gene was amplified by polymerase chain reaction by using K-ras-specific primers followed by mutant enrichment sequencing. Survival differences of patients with a K-ras mutation were compared with those of patients with a normal K-ras status.
RESULTS: A total of 21 patients had a normal K-ras sequence and 14 patients had a K-ras mutation [GAT, n = 7; TGT, n = 3; and GCT, AGT, GTT, GAC (codon 13), n = 1 each]. Median survival of patients with a normal ras sequence from time of treatment with CPT-11 was 332 days compared with 169 days for patients with a K-ras mutation (p = 0.0036). No differences in age, sex, cancer stage, surgical treatment, or chemotherapy treatment were observed.
CONCLUSION: Determination of the presence of a K-ras mutation may predict survival in patients with progressive colon cancer after treatment with 5-fluorouracil who receive CPT-11.

Entities:  

Mesh:

Substances:

Year:  1997        PMID: 9345343     DOI: 10.1097/00000421-199710000-00020

Source DB:  PubMed          Journal:  Am J Clin Oncol        ISSN: 0277-3732            Impact factor:   2.339


  6 in total

1.  FL118, a novel camptothecin analogue, overcomes irinotecan and topotecan resistance in human tumor xenograft models.

Authors:  Xiang Ling; Xiaojun Liu; Kai Zhong; Nicholas Smith; Joshua Prey; Fengzhi Li
Journal:  Am J Transl Res       Date:  2015-10-15       Impact factor: 4.060

2.  Antagonistic effect of flavonoids on NSC-741909-mediated antitumor activity via scavenging of reactive oxygen species.

Authors:  Wei Guo; Xiaoli Wei; Shuhong Wu; Li Wang; Henry Peng; Ji Wang; Bingliang Fang
Journal:  Eur J Pharmacol       Date:  2010-09-18       Impact factor: 4.432

Review 3.  Are RAS mutations predictive markers of resistance to standard chemotherapy?

Authors:  Yohann Loriot; Pierre Mordant; Eric Deutsch; Ken André Olaussen; Jean-Charles Soria
Journal:  Nat Rev Clin Oncol       Date:  2009-07-14       Impact factor: 66.675

4.  KRAS mutation in stage III colon cancer and clinical outcome following intergroup trial CALGB 89803.

Authors:  Shuji Ogino; Jeffrey A Meyerhardt; Natsumi Irahara; Donna Niedzwiecki; Donna Hollis; Leonard B Saltz; Robert J Mayer; Paul Schaefer; Renaud Whittom; Alexander Hantel; Al B Benson; Richard M Goldberg; Monica M Bertagnolli; Charles S Fuchs
Journal:  Clin Cancer Res       Date:  2009-11-24       Impact factor: 12.531

5.  Synthesis of novel 10,11-methylenedioxy-camptothecin glycoside derivatives and investigation of their anti-tumor effects in vivo.

Authors:  Guanzhao Wu; Xiaoyuan Mai; Feng Liu; Mingming Lin; Xueyang Dong; Qingliang Xu; Cui Hao; Lijuan Zhang; Rilei Yu; Tao Jiang
Journal:  RSC Adv       Date:  2019-04-09       Impact factor: 4.036

6.  KRAS and BRAF Mutations as Prognostic and Predictive Biomarkers for Standard Chemotherapy Response in Metastatic Colorectal Cancer: A Single Institutional Study.

Authors:  Nuria Garcia-Carbonero; Javier Martinez-Useros; Weiyao Li; Alberto Orta; Nuria Perez; Cristina Carames; Tatiana Hernandez; Irene Moreno; Gloria Serrano; Jesus Garcia-Foncillas
Journal:  Cells       Date:  2020-01-15       Impact factor: 6.600

  6 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.