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11 in total

1. Synthesis and evaluation of a new series of tri-, di-, and mono-N-alkylcarbamylphloroglucinols as conformationally constrained inhibitors of cholesterol esterase.

Authors: Ming-Cheng Lin; Gin-Zen Lin; Ching-In Hwang; Shuo-Yung Jian; James Lin; Yu-Fong Shen; Gialih Lin
Journal: Protein Sci Date: 2012-08-09 Impact factor: 6.725

2. The First Dual ChE/FAAH Inhibitors: New Perspectives for Alzheimer's Disease?

Authors: Angela Rampa; Manuela Bartolini; Alessandra Bisi; Federica Belluti; Silvia Gobbi; Vincenza Andrisano; Alessia Ligresti; Vincenzo Di Marzo
Journal: ACS Med Chem Lett Date: 2012-01-21 Impact factor: 4.345

3. Stereoselective inhibition of cholesterol esterase by enantiomers of exo- and endo-2-norbornyl-N-n-butylcarbamates.

Authors: Ming-Cheng Lin; Shyh-Jei Yeh; I-Ru Chen; Gialih Lin
Journal: Protein J Date: 2011-03 Impact factor: 2.371

4. Immobilized butyrylcholinesterase in the characterization of new inhibitors that could ease Alzheimer's disease.

Authors: Manuela Bartolini; Nigel H Greig; Qian-Sheng Yu; Vincenza Andrisano
Journal: J Chromatogr A Date: 2008-10-04 Impact factor: 4.759

5. Interaction of the serine hydrolase KIAA1363 with organophosphorus agents: Evaluation of potency and kinetics.

Authors: Matthew K Ross; Kim Pluta; Victoria Bittles; Abdolsamad Borazjani; J Allen Crow
Journal: Arch Biochem Biophys Date: 2015-11-23 Impact factor: 4.013

6. Benzene-di-N-substituted carbamates as conformationally constrained substrate analogs of cholesterol esterase.

Authors: S-Y Chiou; M-C Lin; M-T Hwang; H-G Chang; G Lin
Journal: Protein J Date: 2008-08 Impact factor: 2.371

7. Probing stereoselective inhibition of the acyl binding site of cholesterol esterase with four diastereomers of 2'-N-alpha-methylbenzylcarbamyl-1, 1'-bi-2-naphthol.

Authors: Shyh-Ying Chiou; Cheng-Yue Lai; Long-Yau Lin; Gialih Lin
Journal: BMC Biochem Date: 2005-09-22 Impact factor: 4.059

8. Pharmacophore-based design and discovery of (-)-meptazinol carbamates as dual modulators of cholinesterase and amyloidogenesis.

Authors: Qiong Xie; Zhaoxi Zheng; Biyun Shao; Wei Fu; Zheng Xia; Wei Li; Jian Sun; Wei Zheng; Weiwei Zhang; Wei Sheng; Qihong Zhang; Hongzhuan Chen; Hao Wang; Zhuibai Qiu
Journal: J Enzyme Inhib Med Chem Date: 2017-12 Impact factor: 5.051

9. Inhibition of pancreatic cholesterol esterase reduces cholesterol absorption in the hamster.

Authors: John E Heidrich; Linda M Contos; Lucy A Hunsaker; Lorraine M Deck; David L Vander Jagt
Journal: BMC Pharmacol Date: 2004-04-19

10. Fragment-Sized and Bidentate (Immuno)Proteasome Inhibitors Derived from Cysteine and Threonine Targeting Warheads.

Authors: Levente Kollár; Martina Gobec; Matic Proj; Lara Smrdel; Damijan Knez; Tímea Imre; Ágnes Gömöry; László Petri; Péter Ábrányi-Balogh; Dorottya Csányi; György G Ferenczy; Stanislav Gobec; Izidor Sosič; György M Keserű
Journal: Cells Date: 2021-12-06 Impact factor: 6.600