Literature DB >> 9258348

Synthesis and biology of a 7-nitro-2,1,3-benzoxadiazol-4-yl derivative of 2-phenylindole-3-acetamide: a fluorescent probe for the peripheral-type benzodiazepine receptor.

A P Kozikowski1, M Kotoula, D Ma, N Boujrad, W Tückmantel, V Papadopoulos.   

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Year:  1997        PMID： 9258348     DOI： 10.1021/jm970220w

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  15 in total

Review 1.  Structural and physico-chemical determinants of the interactions of macrocyclic photosensitizers with cells.

Authors:  Halina Mojzisova; Stéphanie Bonneau; Daniel Brault
Journal:  Eur Biophys J       Date:  2007-07-13       Impact factor: 1.733

2.  New structure-activity relationships of N-acetamide substituted pyrazolopyrimidines as pharmacological ligands of TSPO.

Authors:  Jun Li; Michael L Schulte; Michael L Nickels; H Charles Manning
Journal:  Bioorg Med Chem Lett       Date:  2016-06-16       Impact factor: 2.823

3.  New fluorescent probes targeting the mitochondrial-located translocator protein 18 kDa (TSPO) as activated microglia imaging agents.

Authors:  Nunzio Denora; Valentino Laquintana; Adriana Trapani; Hiromi Suzuki; Makoto Sawada; Giuseppe Trapani
Journal:  Pharm Res       Date:  2011-08-05       Impact factor: 4.200

4.  Molecular imaging of the translocator protein (TSPO) in a pre-clinical model of breast cancer.

Authors:  Shelby K Wyatt; H Charles Manning; Mingfeng Bai; Stephanie N Bailey; Pascal Gallant; Guobin Ma; Laura McIntosh; Darryl J Bornhop
Journal:  Mol Imaging Biol       Date:  2009-12-01       Impact factor: 3.488

5.  Development of a unique 3D interaction model of endogenous and synthetic peripheral benzodiazepine receptor ligands.

Authors:  N Cinone; H D Hötje; A Carotti
Journal:  J Comput Aided Mol Des       Date:  2000-11       Impact factor: 3.686

6.  Quantitative, preclinical PET of translocator protein expression in glioma using 18F-N-fluoroacetyl-N-(2,5-dimethoxybenzyl)-2-phenoxyaniline.

Authors:  Jason R Buck; Eliot T McKinley; Matthew R Hight; Allie Fu; Dewei Tang; Ralph Adam Smith; Mohammed Noor Tantawy; Todd E Peterson; Daniel Colvin; Mohammed Sib Ansari; Ronald M Baldwin; Ping Zhao; Saffet Guleryuz; H Charles Manning
Journal:  J Nucl Med       Date:  2010-12-13       Impact factor: 10.057

7.  Pk11195, a mitochondrial benzodiazepine receptor antagonist, reduces apoptosis threshold in Bcl-X(L) and Mcl-1 expressing human cholangiocarcinoma cells.

Authors:  A C Okaro; D A Fennell; M Corbo; B R Davidson; F E Cotter
Journal:  Gut       Date:  2002-10       Impact factor: 23.059

8.  Drug ligand-induced activation of translocator protein (TSPO) stimulates steroid production by aged brown Norway rat Leydig cells.

Authors:  J Y Chung; H Chen; A Midzak; A L Burnett; V Papadopoulos; B R Zirkin
Journal:  Endocrinology       Date:  2013-03-22       Impact factor: 4.736

9.  TSPO targeted dendrimer imaging agent: synthesis, characterization, and cellular internalization.

Authors:  Lynn E Samuelson; Madeline J Dukes; Colette R Hunt; Jonathan D Casey; Darryl J Bornhop
Journal:  Bioconjug Chem       Date:  2009-11       Impact factor: 4.774

Review 10.  Translocator protein 18 kDa (TSPO): molecular sensor of brain injury and repair.

Authors:  Ming-Kai Chen; Tomás R Guilarte
Journal:  Pharmacol Ther       Date:  2008-02-09       Impact factor: 12.310
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