Literature DB >> 9142394

pA, a new scale for the measurement of drug antagonism. 1947.

H O Schild.   

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Year:  1997        PMID： 9142394      PMCID： PMC3224268          DOI： 10.1111/j.1476-5381.1997.tb06773.x

Source DB:  PubMed          Journal:  Br J Pharmacol        ISSN： 0007-1188            Impact factor:   8.739


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  2 in total

1.  A method of conducting a biological assay on a preparation giving repeated graded responses illustrated by the estimation of histamine.

Authors:  H O Schild
Journal:  J Physiol       Date:  1942-06-02       Impact factor: 5.182

2.  Automatic apparatus for pharmacological assays on isolated preparations.

Authors:  H O Schild
Journal:  Br J Pharmacol Chemother       Date:  1946-06
  2 in total
  8 in total

1.  Histamine and antihistamine substances.

Authors:  J H BURN
Journal:  Postgrad Med J       Date:  1948-02       Impact factor: 2.401

2.  Discovery of Polypharmacological Melanocortin-3 and -4 Receptor Probes and Identification of a 100-Fold Selective nM MC3R Agonist versus a μM MC4R Partial Agonist.

Authors:  Katlyn A Fleming; Katie T Freeman; Mike D Powers; Radleigh G Santos; Ginamarie Debevec; Marc A Giulianotti; Richard A Houghten; Skye R Doering; Clemencia Pinilla; Carrie Haskell-Luevano
Journal:  J Med Chem       Date:  2019-02-28       Impact factor: 7.446

3.  Structure-Activity Relationship Studies of a Macrocyclic AGRP-Mimetic Scaffold c[Pro-Arg-Phe-Phe-Asn-Ala-Phe-DPro] Yield Potent and Selective Melanocortin-4 Receptor Antagonists and Melanocortin-5 Receptor Inverse Agonists That Increase Food Intake in Mice.

Authors:  Katlyn A Fleming; Mark D Ericson; Katie T Freeman; Danielle N Adank; Mary M Lunzer; Stacey L Wilber; Carrie Haskell-Luevano
Journal:  ACS Chem Neurosci       Date:  2018-02-13       Impact factor: 4.418

4.  Synergistic Multiresidue Substitutions of a Macrocyclic c[Pro-Arg-Phe-Phe-Asn-Ala-Phe-dPro] Agouti-Related Protein (AGRP) Scaffold Yield Potent and >600-Fold MC4R versus MC3R Selective Melanocortin Receptor Antagonists.

Authors:  Katlyn A Fleming; Katie T Freeman; Mark D Ericson; Carrie Haskell-Luevano
Journal:  J Med Chem       Date:  2018-08-16       Impact factor: 7.446

5.  Modulation by histamine of the delayed outward potassium current in guinea-pig ventricular myocytes.

Authors:  K Yazawa; Y Abiko
Journal:  Br J Pharmacol       Date:  1993-05       Impact factor: 8.739

6.  Delta opioidmimetic antagonists: prototypes for designing a new generation of ultraselective opioid peptides.

Authors:  S Salvadori; M Attila; G Balboni; C Bianchi; S D Bryant; O Crescenzi; R Guerrini; D Picone; T Tancredi; P A Temussi
Journal:  Mol Med       Date:  1995-09       Impact factor: 6.354

7.  Measurement of smooth muscle function in the isolated tissue bath-applications to pharmacology research.

Authors:  Brian Jespersen; Nathan R Tykocki; Stephanie W Watts; Peter J Cobbett
Journal:  J Vis Exp       Date:  2015-01-19       Impact factor: 1.355

8.  Threshold and receptor reserve in the action of neurohypophyseal peptides. A study of synergists and antagonists of the hydroosmotic response of the toad urinary bladder.

Authors:  P Eggena; I L Schwartz; R Walter
Journal:  J Gen Physiol       Date:  1970-08       Impact factor: 4.086
  8 in total

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