Literature DB >> 8765503

Identification of the first retinoid X, receptor homodimer antagonist.

S S Canan Koch1, L J Dardashti, J J Hebert, S K White, G E Croston, K S Flatten, R A Heyman, A M Nadzan.   

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Year:  1996        PMID： 8765503     DOI： 10.1021/jm960311d

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  10 in total

1.  Ligand-dependent degradation of retinoid X receptors does not require transcriptional activity or coactivator interactions.

Authors:  D L Osburn; G Shao; H M Seidel; I G Schulman
Journal:  Mol Cell Biol       Date:  2001-08       Impact factor: 4.272

2.  Spatiotemporal retinoid-X receptor activation detected in live vertebrate embryos.

Authors:  Ayala Luria; J David Furlow
Journal:  Proc Natl Acad Sci U S A       Date:  2004-06-03       Impact factor: 11.205

3.  Coexpression of nuclear receptor partners increases their solubility and biological activities.

Authors:  C Li; J W Schwabe; E Banayo; R M Evans
Journal:  Proc Natl Acad Sci U S A       Date:  1997-03-18       Impact factor: 11.205

4.  Antagonist-perturbation mechanism for activation function-2 fixed motifs: active conformation and docking mode of retinoid X receptor antagonists.

Authors:  Motonori Tsuji
Journal:  J Comput Aided Mol Des       Date:  2017-05-22       Impact factor: 3.686

5.  Nurr1-RXR heterodimers mediate RXR ligand-induced signaling in neuronal cells.

Authors:  Asa Wallen-Mackenzie; Alexander Mata de Urquiza; Susanna Petersson; Francisco J Rodriguez; Stina Friling; Joseph Wagner; Peter Ordentlich; Johan Lengqvist; Richard A Heyman; Ernest Arenas; Thomas Perlmann
Journal:  Genes Dev       Date:  2003-12-17       Impact factor: 11.361

6.  Deuterium exchange and mass spectrometry reveal the interaction differences of two synthetic modulators of RXRalpha LBD.

Authors:  Xuguang Yan; Efrén Pérez; Mark Leid; Michael I Schimerlik; Angel R de Lera; Max L Deinzer
Journal:  Protein Sci       Date:  2007-09-28       Impact factor: 6.725

7.  Modeling, synthesis and biological evaluation of potential retinoid X receptor (RXR) selective agonists: novel analogues of 4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydro-2-naphthyl)ethynyl]benzoic acid (bexarotene).

Authors:  Carl E Wagner; Peter W Jurutka; Pamela A Marshall; Thomas L Groy; Arjan van der Vaart; Joseph W Ziller; Julie K Furmick; Mark E Graeber; Erik Matro; Belinda V Miguel; Ivy T Tran; Jungeun Kwon; Jamie N Tedeschi; Shahram Moosavi; Amina Danishyar; Joshua S Philp; Reina O Khamees; Jevon N Jackson; Darci K Grupe; Syed L Badshah; Justin W Hart
Journal:  J Med Chem       Date:  2009-10-08       Impact factor: 7.446

8.  The "Phantom Effect" of the Rexinoid LG100754: structural and functional insights.

Authors:  Yoshiteru Sato; Nick Ramalanjaona; Tiphaine Huet; Noelle Potier; Judit Osz; Pierre Antony; Carole Peluso-Iltis; Pierre Poussin-Courmontagne; Eric Ennifar; Yves Mély; Annick Dejaegere; Dino Moras; Natacha Rochel
Journal:  PLoS One       Date:  2010-11-30       Impact factor: 3.240

9.  Regulation of RXR-RAR Heterodimers by RXR- and RAR-Specific Ligands and Their Combinations.

Authors:  Albane le Maire; Catherine Teyssier; Patrick Balaguer; William Bourguet; Pierre Germain
Journal:  Cells       Date:  2019-11-05       Impact factor: 6.600

Review 10.  Retinoid X Receptor Antagonists.

Authors:  Masaki Watanabe; Hiroki Kakuta
Journal:  Int J Mol Sci       Date:  2018-08-10       Impact factor: 5.923
  10 in total

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