Literature DB >> 8668667

Effect of change in shape factor of a single crystal on its dissolution behavior.

M V Dali1, J T Carstensen.   

Abstract

PURPOSE: To study the effect of change in the shape factor of real crystals on their dissolution behavior using a potassium dichromate crystal as a model for particulates in general.
METHODS: A model geometry (parallelepiped) has been suggested for a dissolving particle. Single crystals of potassium dichromate which are monoclinic prisms were grown individually from supersaturated solutions at 40 degrees C. Dissolution studies were carried out on five such crystals in 0.1N H2SO4 at 25 degrees C and a stirrer speed of 50 +/- 1 rpm. The five crystals had different degrees of non-isometricity. Initial dimensions of the crystals were measured using image analysis techniques. The shape factor of the dissolving crystal as a function of time was obtained indirectly from the dissolution data.
RESULTS: The shape factor of a single crystal changed significantly after about 50% dissolution. The nature of this change depended on the degree of non-isometricity of the crystal. The change in shape factor of the dissolving crystal was accounted for in the Hixson-Crowell cube root law, and a modified form of the cube root equation was developed. This equation for dissolution explained the observed upward curvature in the cube root law plot.
CONCLUSIONS: The shape factor for any non-isometric particle cannot be considered to be constant over the dissolution event, as is commonly assumed. This change has an appreciable effect on the dissolution behavior of crystals. This study is particularly of significance for elongated shapes like needles and platelets. By the methodology described here, it was possible to determine the initial shape factor of the crystal and the intrinsic dissolution rate constant.

Entities:  

Mesh:

Substances:

Year:  1996        PMID: 8668667     DOI: 10.1023/a:1016010207729

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  12 in total

1.  Sieve cuts as monodisperse powders in dissolution studies.

Authors:  D Brooke
Journal:  J Pharm Sci       Date:  1975-08       Impact factor: 3.534

2.  Nonsink dissolution rate equations.

Authors:  M Patel; J T Carstensen
Journal:  J Pharm Sci       Date:  1975-10       Impact factor: 3.534

3.  Dissolution rates of finely divided drug powders. I. Effect of a distribution of particle sizes in a diffusion-controlled process.

Authors:  W I HIGUCHI; E N HIESTAND
Journal:  J Pharm Sci       Date:  1963-01       Impact factor: 3.534

4.  Dissolution rates of finely divided drug powders. II. Micronized methyl-prednisolone.

Authors:  W I HIGUCHI; E L ROWE; E N HIESTAND
Journal:  J Pharm Sci       Date:  1963-02       Impact factor: 3.534

5.  Theoretical isotropic dissolution of nonspherical particles.

Authors:  P V Pedersen; K F Brown
Journal:  J Pharm Sci       Date:  1976-10       Impact factor: 3.534

6.  Experimental evaluation of three single-particle dissolution models.

Authors:  P V Pedersen; K F Brown
Journal:  J Pharm Sci       Date:  1976-10       Impact factor: 3.534

7.  Nonsink dissolution rate equation.

Authors:  P Pothisiri; J T Carstensen
Journal:  J Pharm Sci       Date:  1973-09       Impact factor: 3.534

8.  Dissolution profile of log-normal powders: exact expression.

Authors:  D Brooke
Journal:  J Pharm Sci       Date:  1973-05       Impact factor: 3.534

9.  Dissolution rate patterns of log-normally distributed powders.

Authors:  J T Carstensen; M N Musa
Journal:  J Pharm Sci       Date:  1972-02       Impact factor: 3.534

10.  Dissolution modeling: factors affecting the dissolution rates of polydisperse powders.

Authors:  A T Lu; M E Frisella; K C Johnson
Journal:  Pharm Res       Date:  1993-09       Impact factor: 4.200

View more
  1 in total

1.  Biorelevant dissolution testing to predict the plasma profile of lipophilic drugs after oral administration.

Authors:  E Nicolaides; M Symillides; J B Dressman; C Reppas
Journal:  Pharm Res       Date:  2001-03       Impact factor: 4.200

  1 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.