Literature DB >> 8308858

A new potent and selective histamine H3 receptor agonist, 4-(1H-imidazol-4-ylmethyl)piperidine.

R C Vollinga1, J P de Koning, F P Jansen, R Leurs, W M Menge, H Timmerman.   

Abstract

Entities:  

Mesh：

Substances：

Year:  1994        PMID： 8308858     DOI： 10.1021/jm00029a002

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


× No keyword cloud information.
  11 in total

1.  Interaction Between Brain Histamine and Serotonin, Norepinephrine, and Dopamine Systems: In Vivo Microdialysis and Electrophysiology Study.

Authors:  Gunnar Flik; Joost H A Folgering; Thomas I H F Cremers; Ben H C Westerink; Eliyahu Dremencov
Journal:  J Mol Neurosci       Date:  2015-03-29       Impact factor: 3.444

Review 2.  An update on histamine H3 receptors and gastrointestinal functions.

Authors:  G Bertaccini; G Coruzzi
Journal:  Dig Dis Sci       Date:  1995-09       Impact factor: 3.199

Review 3.  H3 receptors and pain modulation: peripheral, spinal, and brain interactions.

Authors:  Lindsay B Hough; Frank L Rice
Journal:  J Pharmacol Exp Ther       Date:  2010-09-23       Impact factor: 4.030

4.  Inhibition of cortical acetylcholine release and cognitive performance by histamine H3 receptor activation in rats.

Authors:  P Blandina; M Giorgetti; L Bartolini; M Cecchi; H Timmerman; R Leurs; G Pepeu; M G Giovannini
Journal:  Br J Pharmacol       Date:  1996-12       Impact factor: 8.739

Review 5.  International Union of Basic and Clinical Pharmacology. XCVIII. Histamine Receptors.

Authors:  Pertti Panula; Paul L Chazot; Marlon Cowart; Ralf Gutzmer; Rob Leurs; Wai L S Liu; Holger Stark; Robin L Thurmond; Helmut L Haas
Journal:  Pharmacol Rev       Date:  2015-07       Impact factor: 25.468

6.  Activation of peripheral and spinal histamine H3 receptors inhibits formalin-induced inflammation and nociception, respectively.

Authors:  Keri E Cannon; Rob Leurs; Lindsay B Hough
Journal:  Pharmacol Biochem Behav       Date:  2007-07-25       Impact factor: 3.533

7.  Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5-HT3 receptor revealed.

Authors:  R Leurs; M T Tulp; W M Menge; M J Adolfs; O P Zuiderveld; H Timmerman
Journal:  Br J Pharmacol       Date:  1995-10       Impact factor: 8.739

8.  Characterization of the binding of the first selective radiolabelled histamine H3-receptor antagonist, [125I]-iodophenpropit, to rat brain.

Authors:  F P Jansen; T S Wu; H P Voss; H W Steinbusch; R C Vollinga; B Rademaker; A Bast; H Timmerman
Journal:  Br J Pharmacol       Date:  1994-10       Impact factor: 8.739

9.  Cardiovascular effects of selective agonists and antagonists of histamine H3 receptors in the anaesthetized rat.

Authors:  G Coruzzi; E Gambarelli; G Bertaccini; H Timmerman
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1995-06       Impact factor: 3.000

10.  Identification and characterization of ZEL-H16 as a novel agonist of the histamine H3 receptor.

Authors:  Ying Shi; Rong Sheng; Tingting Zhong; Yu Xu; Xiaopan Chen; Dong Yang; Yi Sun; Fenyan Yang; Yongzhou Hu; Naiming Zhou
Journal:  PLoS One       Date:  2012-08-01       Impact factor: 3.240
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.