Warning: Undefined array key "mm" in /www/wwwroot/www.ai-bt.com/si.php on line 10 Deprecated: trim(): Passing null to parameter #1 ($string) of type string is deprecated in /www/wwwroot/www.ai-bt.com/si.php on line 10 Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential.

× No keyword cloud information.

17 in total

1. Immune enhancing effects of dehydroepiandrosterone and dehydroepiandrosterone sulphate and the role of steroid sulphatase.

Authors: A J Suitters; S Shaw; M R Wales; J P Porter; J Leonard; R Woodger; H Brand; M Bodmer; R Foulkes
Journal: Immunology Date: 1997-06 Impact factor: 7.397

2. Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health.

Authors: Mark P Thomas; Barry V L Potter
Journal: J Med Chem Date: 2015-06-12 Impact factor: 7.446

3. Synthesis and evaluation of general mechanism-based inhibitors of sulfatases based on (difluoro)methyl phenyl sulfate and cyclic phenyl sulfamate motifs.

Authors: Sarah R Hanson; Lisa J Whalen; Chi-Huey Wong
Journal: Bioorg Med Chem Date: 2006-10-11 Impact factor: 3.641

4. The effect of the steroid sulfatase inhibitor (p-O-sulfamoyl)-tetradecanoyl tyramine (DU-14) on learning and memory in rats with selective lesion of septal-hippocampal cholinergic tract.

Authors: P A Babalola; N F Fitz; R B Gibbs; P T Flaherty; P-K Li; D A Johnson
Journal: Neurobiol Learn Mem Date: 2012-09-26 Impact factor: 2.877

5. C-3- and C-4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors.

Authors: Dharshini Ganeshapillai; L W Lawrence Woo; Mark P Thomas; Atul Purohit; Barry V L Potter
Journal: ACS Omega Date: 2018-09-06

Review 6. Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: structure-function studies and inhibitor development.

Authors: Yanyan Hong; Shiuan Chen
Journal: Mol Cell Endocrinol Date: 2010-10-01 Impact factor: 4.102

7. Proton-in-flight mechanism for the spontaneous hydrolysis of N-methyl O-phenyl sulfamate: implications for the design of steroid sulfatase inhibitors.

Authors: David R Edwards; Richard Wolfenden
Journal: J Org Chem Date: 2012-04-18 Impact factor: 4.354

Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential.