Literature DB >> 8268120

Local myotoxicity of bupivacaine in rabbits after continuous supraclavicular brachial plexus block.

P Pere1, H Watanabe, M Pitkänen, T Wahlström, P H Rosenberg.   

Abstract

BACKGROUND AND OBJECTIVES: Local anesthetics including bupivacaine have been known to be myotoxic. Continuous brachial plexus blocks with bupivacaine provide good postoperative pain relief, but their effects on the surrounding muscles have not been studied.
METHODS: Eight rabbits were given continuous bilateral brachial plexus blocks with 0.25% bupivacaine (BUPI) and another eight (SALINE) equivalent volumes of saline infused into the plexus region under pentobarbital-ketamine sedation. At the end of the 24-hour blocks, muscle biopsies were taken from one side of the neck in both groups. A week later, the biopsy procedure was repeated on the other side. Plasma concentrations of bupivacaine were measured before and at the end of the 24-hour blocks.
RESULTS: Inflammatory cell infiltration and muscle fiber necrosis were significantly more common in the BUPI than in the SALINE group (p < 0.001). At the end of the continuous block, predominantly neutrophils were found, but in the BUPI group large amounts of eosinophilic granulocytes also were found. A week later lymphocytes, plasma cells, macrophages, and fibroblasts were seen as a sign of beginning scar formation. Plasma concentrations of bupivacaine at 24 hours were at a nontoxic level (0.28-0.71 microgram/ml).
CONCLUSIONS: Brachial plexus blocks with bupivacaine caused reversible myotoxicity and inflammation in the rabbit. A week after the continuous blocks, muscle fiber regeneration had already started.

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Year:  1993        PMID: 8268120

Source DB:  PubMed          Journal:  Reg Anesth        ISSN: 0146-521X


  15 in total

Review 1.  [Toxicology of local anesthetics. Clinical, therapeutic and pathological mechanisms].

Authors:  W Zink; B M Graf
Journal:  Anaesthesist       Date:  2003-12       Impact factor: 1.041

2.  An ultrasound-guided technique for axillary brachial plexus nerve block in rabbits.

Authors:  Carla Fonseca; Anna Server; Marielle Esteves; David Barastegui; Marta Rosal; Cesar G Fontecha; Francisco Soldado
Journal:  Lab Anim (NY)       Date:  2015-05       Impact factor: 12.625

3.  Multivesicular liposomal bupivacaine at the sciatic nerve.

Authors:  J Brian McAlvin; Robert F Padera; Sahadev A Shankarappa; Gally Reznor; Albert H Kwon; Homer H Chiang; Jason Yang; Daniel S Kohane
Journal:  Biomaterials       Date:  2014-03-06       Impact factor: 12.479

4.  Prolonged Duration Local Anesthesia Using Liposomal Bupivacaine Combined With Liposomal Dexamethasone and Dexmedetomidine.

Authors:  Alina Y Rwei; Robert T Sherburne; David Zurakowski; Bruce Wang; Daniel S Kohane
Journal:  Anesth Analg       Date:  2018-04       Impact factor: 5.108

5.  Perineural dexmedetomidine added to ropivacaine causes a dose-dependent increase in the duration of thermal antinociception in sciatic nerve block in rat.

Authors:  Chad M Brummett; Amrita K Padda; Francesco S Amodeo; Kathleen B Welch; Ralph Lydic
Journal:  Anesthesiology       Date:  2009-11       Impact factor: 7.892

6.  Local myotoxicity from sustained release of bupivacaine from microparticles.

Authors:  Robert Padera; Evangelia Bellas; Julie Y Tse; Daphne Hao; Daniel S Kohane
Journal:  Anesthesiology       Date:  2008-05       Impact factor: 7.892

Review 7.  Evaluation of treatments for myofascial pain syndrome and fibromyalgia.

Authors:  Nathan J Rudin
Journal:  Curr Pain Headache Rep       Date:  2003-12

8.  Prolonged duration local anesthesia with minimal toxicity.

Authors:  Hila Epstein-Barash; Iris Shichor; Albert H Kwon; Sherwood Hall; Michael W Lawlor; Robert Langer; Daniel S Kohane
Journal:  Proc Natl Acad Sci U S A       Date:  2009-04-13       Impact factor: 11.205

9.  Perineural administration of dexmedetomidine in combination with bupivacaine enhances sensory and motor blockade in sciatic nerve block without inducing neurotoxicity in rat.

Authors:  Chad M Brummett; Mary A Norat; John M Palmisano; Ralph Lydic
Journal:  Anesthesiology       Date:  2008-09       Impact factor: 7.892

10.  Local toxicity from local anesthetic polymeric microparticles.

Authors:  J Brian McAlvin; Gally Reznor; Sahadev A Shankarappa; Cristina F Stefanescu; Daniel S Kohane
Journal:  Anesth Analg       Date:  2013-03-04       Impact factor: 5.108

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