Literature DB >> 8182696

3'-(Arylmethyl)- and 3'-(aryloxy)-3-phenyl-4-hydroxyquinolin-2(1H)-ones: orally active antagonists of the glycine site on the NMDA receptor.

J J Kulagowski1, R Baker, N R Curtis, P D Leeson, I M Mawer, A M Moseley, M P Ridgill, M Rowley, I Stansfield, A C Foster.   

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Year:  1994        PMID： 8182696     DOI： 10.1021/jm00036a002

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  7 in total

1.  Synthesis and Biological Evaluation of Novel Multi-target-Directed Benzazepines Against Excitotoxicity.

Authors:  Jatin Machhi; Navnit Prajapati; Ashutosh Tripathi; Zalak S Parikh; Ashish M Kanhed; Kirti Patel; Prakash P Pillai; Rajani Giridhar; Mange Ram Yadav
Journal:  Mol Neurobiol       Date:  2016-10-15       Impact factor: 5.590

2.  Synthesis and Biological Screening of Pyrano[3,2-c]quinoline Analogues as Anti-inflammatory and Anticancer Agents.

Authors:  Kuldip D Upadhyay; Narsinh M Dodia; Rupesh C Khunt; Ravi S Chaniara; Anamik K Shah
Journal:  ACS Med Chem Lett       Date:  2018-02-23       Impact factor: 4.345

3.  Inhibition of cortical spreading depression by L-701,324, a novel antagonist at the glycine site of the N-methyl-D-aspartate receptor complex.

Authors:  T P Obrenovitch; E Zilkha
Journal:  Br J Pharmacol       Date:  1996-03       Impact factor: 8.739

Review 4.  Carboxylic acid (bio)isosteres in drug design.

Authors:  Carlo Ballatore; Donna M Huryn; Amos B Smith
Journal:  ChemMedChem       Date:  2013-01-29       Impact factor: 3.466

5.  Molecular electrostatic potentials in aromatic substituted 4-hydroxyquino-2-lones: glycine/NMDA receptor antagonists.

Authors:  Kaustubh A Joshi; Dinannath D Patil; Shridhar P Gejji
Journal:  J Mol Model       Date:  2008-12-09       Impact factor: 1.810

6.  Effects of a partial agonist and a full antagonist acting at the glycine site of the NMDA receptor on inflammation-induced mechanical hyperalgesia in rats.

Authors:  J M Laird; G S Mason; J Webb; R G Hill; R J Hargreaves
Journal:  Br J Pharmacol       Date:  1996-04       Impact factor: 8.739

Review 7.  Development of PET and SPECT probes for glutamate receptors.

Authors:  Takeshi Fuchigami; Morio Nakayama; Sakura Yoshida
Journal:  ScientificWorldJournal       Date:  2015-03-22
  7 in total

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