Literature DB >> 8057295

GABAA receptor agonists, partial agonists, and antagonists. Design and therapeutic prospects.

P Krogsgaard-Larsen1, B Frølund, F S Jørgensen, A Schousboe.   

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Year:  1994        PMID: 8057295     DOI: 10.1021/jm00042a001

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


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  12 in total

1.  Distinct activities of GABA agonists at synaptic- and extrasynaptic-type GABAA receptors.

Authors:  Martin Mortensen; Bjarke Ebert; Keith Wafford; Trevor G Smart
Journal:  J Physiol       Date:  2010-02-22       Impact factor: 5.182

2.  5-tert-Butyl-2-(4'-[18F]fluoropropynylphenyl)-1,3-dithiane oxides: potential new GABA A receptor radioligands.

Authors:  Xuehe Li; Yong-Woon Jung; Scott E Snyder; Joseph Blair; Philip S Sherman; Timothy Desmond; Kirk A Frey; Michael R Kilbourn
Journal:  Nucl Med Biol       Date:  2007-11-26       Impact factor: 2.408

3.  Molecular modelling and conformational analysis of a GABAB antagonist.

Authors:  B Pirard; F Durant
Journal:  J Comput Aided Mol Des       Date:  1996-02       Impact factor: 3.686

4.  GABA is a modulator, rather than a classical transmitter, in the medial nucleus of the trapezoid body-lateral superior olive sound localization circuit.

Authors:  Alexander U Fischer; Nicolas I C Müller; Thomas Deller; Domenico Del Turco; Jonas O Fisch; Désirée Griesemer; Kathrin Kattler; Ayse Maraslioglu; Vera Roemer; Matthew A Xu-Friedman; Jörn Walter; Eckhard Friauf
Journal:  J Physiol       Date:  2019-03-12       Impact factor: 5.182

5.  Neurotoxicity of lindane and picrotoxin: neurochemical and electrophysiological correlates in the rat hippocampus in vivo.

Authors:  Gabriella Nyitrai; Katalin A Kékesi; Nóra Szilágyi; Andrea Papp; Gábor Juhász; Julianna Kardos
Journal:  Neurochem Res       Date:  2002-02       Impact factor: 3.996

6.  Reciprocal innervation between serotonergic and GABAergic neurons in raphe nuclei of the rat.

Authors:  E Bagdy; I Kiraly; L G Harsing
Journal:  Neurochem Res       Date:  2000-11       Impact factor: 3.996

7.  Intestinal gaboxadol absorption via PAT1 (SLC36A1): modified absorption in vivo following co-administration of L-tryptophan.

Authors:  M Larsen; R Holm; K G Jensen; B Brodin; C U Nielsen
Journal:  Br J Pharmacol       Date:  2009-07-07       Impact factor: 8.739

Review 8.  The diversity of GABAA receptors. Pharmacological and electrophysiological properties of GABAA channel subtypes.

Authors:  W Hevers; H Lüddens
Journal:  Mol Neurobiol       Date:  1998-08       Impact factor: 5.590

9.  Synthesis of GABAA receptor agonists and evaluation of their alpha-subunit selectivity and orientation in the GABA binding site.

Authors:  Michaela Jansen; Holger Rabe; Axelle Strehle; Sandra Dieler; Fabian Debus; Gerd Dannhardt; Myles H Akabas; Hartmut Lüddens
Journal:  J Med Chem       Date:  2008-07-24       Impact factor: 7.446

10.  The pharmacology of the neurochemical transmission in the midbrain raphe nuclei of the rat.

Authors:  L G Harsing
Journal:  Curr Neuropharmacol       Date:  2006-10       Impact factor: 7.363

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