Literature DB >> 8057272

Evolution of a novel series of [(N,N-dimethylamino)propyl]- and piperazinylbenzanilides as the first selective 5-HT1D antagonists.

J W Clitherow1, D I Scopes, M Skingle, C C Jordan, W Feniuk, I B Campbell, M C Carter, E W Collington, H E Connor, G A Higgins.   

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Year:  1994        PMID： 8057272     DOI： 10.1021/jm00041a001

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  12 in total

1.  5-HT-stimulated [35S]guanosine-5'-O-(3-thio)triphosphate binding as an assay for functional activation of G proteins coupled with 5-HT1B receptors in rat striatal membranes.

Authors:  Yuji Odagaki; Ryoichi Toyoshima
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2006-02-21       Impact factor: 3.000

2.  Pharmacological evidence that alpha1-and alpha2-adrenoceptors mediate vasoconstriction of carotid arteriovenous anastomoses in anaesthetized pigs.

Authors:  E W Willems; M Trion; P De Vries; J P Heiligers; C M Villalón; P R Saxena
Journal:  Br J Pharmacol       Date:  1999-07       Impact factor: 8.739

3.  Functional characterization and m-RNA expression of 5-HT receptors mediating contraction in human umbilical artery.

Authors:  F Lovren; X F Li; J Lytton; C Triggle
Journal:  Br J Pharmacol       Date:  1999-07       Impact factor: 8.739

4.  Influence of the endothelium and nitric oxide on the contractile responses evoked by 5-HT1D receptor agonists in the rabbit isolated saphenous vein.

Authors:  J P Valentin; R Bonnafous; G W John
Journal:  Br J Pharmacol       Date:  1996-09       Impact factor: 8.739

5.  Investigation of the role of 5-HT1B and 5-HT1D receptors in the sumatriptan-induced constriction of porcine carotid arteriovenous anastomoses.

Authors:  P De Vries; E W Willems; J P Heiligers; C M Villalón; P R Saxena
Journal:  Br J Pharmacol       Date:  1999-05       Impact factor: 8.739

6.  Influence of the 5-HT(2C) receptor antagonist SB242,084 on behaviour produced by the 5-HT(2) agonist Ro60-0175 and the indirect 5-HT agonist dexfenfluramine.

Authors:  G A Higgins; A M Ouagazzal; A J Grottick
Journal:  Br J Pharmacol       Date:  2001-06       Impact factor: 8.739

7.  Functional serotonin 5-HT1D receptors and 5-HT1D beta receptor mRNA expression in human umbilical vein endothelial cells.

Authors:  P Schoeffter; C Ullmer; M Gutierrez; G Weitz-Schmidt; H Lübbert
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1995-11       Impact factor: 3.000

8.  Promotion of cell growth by stimulation of cloned human 5-HT1D receptor sites in transfected C6-glial cells is highly sensitive to intrinsic activity at 5-HT1D receptors.

Authors:  P J Pauwels; T Wurch; C Palmier; F C Colpaert
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1996-07       Impact factor: 3.000

9.  5-Hydroxytryptamine 5-HT1D receptors mediating inhibition of cyclic AMP accumulation in Madin-Darby canine kidney (MDCK) cells.

Authors:  P Schoeffter; I Bobirnac
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1995-09       Impact factor: 3.000

10.  Sumatriptan-induced saphenous venoconstriction in the anaesthetized dog through 5-HT1-like receptor activation.

Authors:  C Drieu la Rochelle; S E O'Connor
Journal:  Br J Pharmacol       Date:  1995-10       Impact factor: 8.739
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