Literature DB >> 7699699

N-(1-methyl-5-indolyl)-N'-(3-methyl-5-isothiazolyl)urea: a novel, high-affinity 5-HT2B receptor antagonist.

I T Forbes1, G E Jones, O E Murphy, V Holland, G S Baxter.   

Abstract

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Year:  1995        PMID： 7699699     DOI： 10.1021/jm00006a001

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  17 in total

1.  Evidence that activation of central 5-HT(2B) receptors causes renal sympathoexcitation in anaesthetized rats.

Authors:  I D Knowles; A G Ramage
Journal:  Br J Pharmacol       Date:  2000-01       Impact factor: 8.739

2.  Smooth muscle 5-HT2A receptors mediating contraction of porcine isolated proximal stomach strips.

Authors:  P Janssen; N H Prins; A L Meulemans; R A Lefebvre
Journal:  Br J Pharmacol       Date:  2002-12       Impact factor: 8.739

3.  Serotonin modulates the population activity profile of olfactory bulb external tufted cells.

Authors:  Shaolin Liu; Jason L Aungst; Adam C Puche; Michael T Shipley
Journal:  J Neurophysiol       Date:  2011-10-19       Impact factor: 2.714

4.  RS-127445: a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist.

Authors:  D W Bonhaus; L A Flippin; R J Greenhouse; S Jaime; C Rocha; M Dawson; K Van Natta; L K Chang; T Pulido-Rios; A Webber; E Leung; R M Eglen; G R Martin
Journal:  Br J Pharmacol       Date:  1999-07       Impact factor: 8.739

5.  Contribution of serotonin (5-HT) 5-HT2 receptor subtypes to the discriminative stimulus effects of cocaine in rats.

Authors:  Malgorzata Filip; Marcy J Bubar; Kathryn A Cunningham
Journal:  Psychopharmacology (Berl)       Date:  2005-10-28       Impact factor: 4.530

6.  Characterization of the receptors involved in the 5-HT-induced excitation of canine antral longitudinal muscle.

Authors:  N H Prins; L M Akkermans; R A Lefebvre; J A Schuurkes
Journal:  Br J Pharmacol       Date:  2001-11       Impact factor: 8.739

7.  Contractile effects of 5-hydroxytryptamine and 5-carboxamidotryptamine in the equine jejunum.

Authors:  Cathérine Delesalle; Piet Deprez; Jan A J Schuurkes; Romain A Lefebvre
Journal:  Br J Pharmacol       Date:  2006-01       Impact factor: 8.739

8.  Evidence for a role for central 5-HT2B as well as 5-HT2A receptors in cardiovascular regulation in anaesthetized rats.

Authors:  I D Knowles; A G Ramage
Journal:  Br J Pharmacol       Date:  1999-10       Impact factor: 8.739

9.  Functional 5-HT receptors in human occipital artery.

Authors:  Raphaela Verheggen; Andreas Meier; Inga Werner; Andreas Wienekamp; Thomas Kruschat; Trond Brattelid; Finn Olav Levy; Alberto Kaumann
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2004-03-06       Impact factor: 3.000

10.  5-HT(2B) antagonism arrests non-canonical TGF-β1-induced valvular myofibroblast differentiation.

Authors:  Joshua D Hutcheson; Larisa M Ryzhova; Vincent Setola; W David Merryman
Journal:  J Mol Cell Cardiol       Date:  2012-08-23       Impact factor: 5.000
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