Literature DB >> 7541854

Placebo controlled double-blind study to test the efficacy of the aromatase inhibitor atamestane in patients with benign prostatic hyperplasia not requiring operation. The Schering 90.062 Study Group.

J C Gingell1, H Knönagel, K H Kurth, U W Tunn.   

Abstract

PURPOSE: We tested the theoretical concept that a selective decrease in estrogens has a beneficial therapeutic effect on established benign prostatic hyperplasia.
MATERIALS AND METHODS: In a double-blind study 160 patients from 14 centers were randomized between 2 groups to receive either placebo or the aromatase inhibitor atamestane (1-methyl-androsin-1,4 diene-3 17-dione, 400 mg. daily for 48 weeks).
RESULTS: The aromatase inhibitor decreased the mean estradiol level by approximately 40% and estrone by 60%. The testosterone concentration increased by more than 40% and dihydrotestosterone increased to 30%. Analysis of clinical parameters showed no difference between placebo and atamestane.
CONCLUSIONS: The counter regulatory increase in androgens may counterbalance any positive effect of the decrease in estrogens to preserve intraprostatic homeostasis.

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Year:  1995        PMID: 7541854     DOI: 10.1097/00005392-199508000-00020

Source DB:  PubMed          Journal:  J Urol        ISSN: 0022-5347            Impact factor:   7.450


  5 in total

1.  Best of the 2004 AUA Annual Meeting: Highlights from the 2004 Annual Meeting of the American Urological Association, May 8-13, 2004, San Francisco, CA.

Authors: 
Journal:  Rev Urol       Date:  2004

Review 2.  Androgens and estrogens in benign prostatic hyperplasia: past, present and future.

Authors:  Tristan M Nicholson; William A Ricke
Journal:  Differentiation       Date:  2011-05-26       Impact factor: 3.880

Review 3.  Expanding the therapeutic use of androgens via selective androgen receptor modulators (SARMs).

Authors:  Wenqing Gao; James T Dalton
Journal:  Drug Discov Today       Date:  2007-02-07       Impact factor: 7.851

4.  Toremifene-atamestane; alone or in combination: predictions from the preclinical intratumoral aromatase model.

Authors:  Gauri J Sabnis; Luciana Macedo; Olga Goloubeva; Adam Schayowitz; Yue Zhu; Angela Brodie
Journal:  J Steroid Biochem Mol Biol       Date:  2007-09-07       Impact factor: 4.292

Review 5.  Dehydroepiandrosterone: a potential therapeutic agent in the treatment and rehabilitation of the traumatically injured patient.

Authors:  Conor Bentley; Jon Hazeldine; Carolyn Greig; Janet Lord; Mark Foster
Journal:  Burns Trauma       Date:  2019-08-02
  5 in total

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