Literature DB >> 7495678

Design and pharmacology of peptide mimetics.

G J Moore1, J R Smith, B W Baylis, J M Matsoukas.   

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Year:  1995        PMID: 7495678     DOI: 10.1016/s1054-3589(08)60667-5

Source DB:  PubMed          Journal:  Adv Pharmacol        ISSN: 1054-3589


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  7 in total

1.  An efficient synthesis of a rationally designed 1,5 disubstituted imidazole AT(1) angiotensin II receptor antagonist: reorientation of imidazole pharmacophore groups in losartan reserves high receptor affinity and confirms docking studies.

Authors:  George Agelis; Panagiota Roumelioti; Amalia Resvani; Serdar Durdagi; Maria-Eleni Androutsou; Konstantinos Kelaidonis; Demetrios Vlahakos; Thomas Mavromoustakos; John Matsoukas
Journal:  J Comput Aided Mol Des       Date:  2010-07-10       Impact factor: 3.686

2.  Hinge peptide combinatorial libraries for inhilbitors of botulinum neurotoxins and saxitoxin: deconvolution strategy.

Authors:  Graham J Moore; Diana M Moore; Samir S Roy; Lawrence J Hayden; Murray G Hamilton; Nora W C Chan; William E Lee
Journal:  Mol Divers       Date:  2006-02       Impact factor: 2.943

3.  Understanding the Driving Forces That Trigger Mutations in SARS-CoV-2: Mutational Energetics and the Role of Arginine Blockers in COVID-19 Therapy.

Authors:  Harry Ridgway; Christos T Chasapis; Konstantinos Kelaidonis; Irene Ligielli; Graham J Moore; Laura Kate Gadanec; Anthony Zulli; Vasso Apostolopoulos; Thomas Mavromoustakos; John M Matsoukas
Journal:  Viruses       Date:  2022-05-11       Impact factor: 5.818

4.  A tree-based algorithm for determining the effects of solvation on the structure of salivary gland tripeptide NH3+-D-PHE-D-GLU-GLY-COO-.

Authors:  Essam Metwally; Heba A Ismail; Joseph S Davison; Ronald Mathison
Journal:  Biophys J       Date:  2003-09       Impact factor: 4.033

Review 5.  A Global Review on Short Peptides: Frontiers and Perspectives.

Authors:  Vasso Apostolopoulos; Joanna Bojarska; Tsun-Thai Chai; Sherif Elnagdy; Krzysztof Kaczmarek; John Matsoukas; Roger New; Keykavous Parang; Octavio Paredes Lopez; Hamideh Parhiz; Conrad O Perera; Monica Pickholz; Milan Remko; Michele Saviano; Mariusz Skwarczynski; Yefeng Tang; Wojciech M Wolf; Taku Yoshiya; Janusz Zabrocki; Piotr Zielenkiewicz; Maha AlKhazindar; Vanessa Barriga; Konstantinos Kelaidonis; Elham Mousavinezhad Sarasia; Istvan Toth
Journal:  Molecules       Date:  2021-01-15       Impact factor: 4.411

Review 6.  From Angiotensin II to Cyclic Peptides and Angiotensin Receptor Blockers (ARBs): Perspectives of ARBs in COVID-19 Therapy.

Authors:  John Matsoukas; Vasso Apostolopoulos; Anthony Zulli; Graham Moore; Konstantinos Kelaidonis; Kalliopi Moschovou; Thomas Mavromoustakos
Journal:  Molecules       Date:  2021-01-25       Impact factor: 4.411

7.  Discovery of a new generation of angiotensin receptor blocking drugs: Receptor mechanisms and in silico binding to enzymes relevant to SARS-CoV-2.

Authors:  Harry Ridgway; Graham J Moore; Thomas Mavromoustakos; Sotirios Tsiodras; Irene Ligielli; Konstantinos Kelaidonis; Christos T Chasapis; Laura Kate Gadanec; Anthony Zulli; Vasso Apostolopoulos; Russell Petty; Ioannis Karakasiliotis; Vassilis G Gorgoulis; John M Matsoukas
Journal:  Comput Struct Biotechnol J       Date:  2022-04-09       Impact factor: 6.155

  7 in total

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