Literature DB >> 7494855

Molecular pharmacological aspects of histamine receptors.

R Leurs1, M J Smit, H Timmerman.   

Abstract

In this article, we review the recent developments in the field of histamine research. Besides the description of pharmacological tools for the H1, H2 and H3 receptor, specific attention is paid to both the molecular aspects of the receptor proteins, including the recent cloning of the receptor genes, and their respective signal transduction mechanisms.

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Year:  1995        PMID： 7494855     DOI： 10.1016/0163-7258(95)00006-3

Source DB:  PubMed          Journal:  Pharmacol Ther        ISSN： 0163-7258            Impact factor:   12.310


  54 in total

1.  Modulation of histamine H(2) receptor signalling by G-protein-coupled receptor kinase 2 and 3.

Authors:  M S Rodriguez-Pena; H Timmerman; R Leurs
Journal:  Br J Pharmacol       Date:  2000-12       Impact factor: 8.739

Review 2.  New insights into the second generation antihistamines.

Authors:  G M Walsh; L Annunziato; N Frossard; K Knol; S Levander; J M Nicolas; M Taglialatela; M D Tharp; J P Tillement; H Timmerman
Journal:  Drugs       Date:  2001       Impact factor: 9.546

3.  Effect of histamine on spontaneous contractions of mesenteric lymphatic vessels and lymph nodes of white rats: endothelium-dependent responses.

Authors:  S G Petunov; A A Egorova; R S Orlov; E R Nikitina
Journal:  Dokl Biol Sci       Date:  2010-06-22

4.  Inverse agonism of histamine H2 antagonist accounts for upregulation of spontaneously active histamine H2 receptors.

Authors:  M J Smit; R Leurs; A E Alewijnse; J Blauw; G P Van Nieuw Amerongen; Y Van De Vrede; E Roovers; H Timmerman
Journal:  Proc Natl Acad Sci U S A       Date:  1996-06-25       Impact factor: 11.205

5.  Histamine H(3) receptor-mediated inhibition of depolarization-induced, dopamine D(1) receptor-dependent release of [(3)H]-gamma-aminobutryic acid from rat striatal slices.

Authors:  J A Arias-Montaño; B Floran; M Garcia; J Aceves; J M Young
Journal:  Br J Pharmacol       Date:  2001-05       Impact factor: 8.739

6.  Safety, tolerability and pharmacokinetics of the histamine H3 receptor antagonist, ABT-288, in healthy young adults and elderly volunteers.

Authors:  Ahmed A Othman; George Haig; Hana Florian; Charles Locke; Jun Zhang; Sandeep Dutta
Journal:  Br J Clin Pharmacol       Date:  2013-05       Impact factor: 4.335

7.  Targeted disruption of H3 receptors results in changes in brain histamine tone leading to an obese phenotype.

Authors:  Kazuhiko Takahashi; Hiroaki Suwa; Tomoo Ishikawa; Hidehito Kotani
Journal:  J Clin Invest       Date:  2002-12       Impact factor: 14.808

8.  Effects of histamine on the contractile and electrical activity in isolated lymphatic vessels of the guinea-pig mesentery.

Authors:  James L R Fox; Pierre-Yves von der Weid
Journal:  Br J Pharmacol       Date:  2002-08       Impact factor: 8.739

9.  Cytokine responses of intraepithelial lymphocytes are regulated by histamine H(2) receptor.

Authors:  Kosuke Takagaki; Satoshi Osawa; Yoshiaki Horio; Takanori Yamada; Yasushi Hamaya; Yasuhiro Takayanagi; Takahisa Furuta; Akira Hishida; Mutsuhiro Ikuma
Journal:  J Gastroenterol       Date:  2009-03-10       Impact factor: 7.527

10.  Histamine H(3) receptor-mediated signaling protects mice from cerebral malaria.

Authors:  Walid Beghdadi; Adeline Porcherie; Bradley S Schneider; Séverine Morisset; David Dubayle; Roger Peronet; Michel Dy; Jacques Louis; Jean-Michel Arrang; Salaheddine Mécheri
Journal:  PLoS One       Date:  2009-06-23       Impact factor: 3.240
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