Literature DB >> 7398762

Histamine H1-receptors labeled in vivo: antidepressant and antihistamine interactions.

D Diffley, V T Tran, S H Snyder.   

Abstract

3H-Mepyramine labels specific histamine H1-receptors in brains of mice after intravenous injection. The potencies of H1-antihistamines in reducing 3H-mepyramine binding in vivo correspond to their pharmacological activities and show parallels with their affinities for 3H-mepyramine binding sites in isolated brain membranes. Several antidepressants are potent in competing for 3H-mepyramine binding in vivo as well as in vitro.

Entities:  

Mesh：

Substances：

Year:  1980        PMID： 7398762     DOI： 10.1016/0014-2999(80)90043-6

Source DB:  PubMed          Journal:  Eur J Pharmacol        ISSN： 0014-2999            Impact factor:   4.432


  6 in total

1.  H1-receptor antagonists: comparative pharmacology and clinical use.

Authors:  D Reinhardt; U Borchard
Journal:  Klin Wochenschr       Date:  1982-09-01

2.  Acceleration of rat brain beta-adrenoceptor subsensitivity following the coadministration of histamine receptor antagonists with imipramine.

Authors:  A A Alhaider; A A Mustafa
Journal:  Agents Actions       Date:  1989-11

3.  Histamine levels and clonic convulsions of electrically-induced seizure in mice: the effects of alpha-fluoromethylhistidine and metoprine.

Authors:  H Yokoyama; K Onodera; K Maeyama; K Yanai; K Iinuma; L Tuomisto; T Watanabe
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1992-07       Impact factor: 3.000

4.  Alteration of histamine metabolism in the rat brain under influence of various antidepressive treatments.

Authors:  J Zawilska; J Z Nowak
Journal:  Agents Actions       Date:  1985-04

5.  Histamine H1 receptor occupancy in human brains after single oral doses of histamine H1 antagonists measured by positron emission tomography.

Authors:  K Yanai; J H Ryu; T Watanabe; R Iwata; T Ido; Y Sawai; K Ito; M Itoh
Journal:  Br J Pharmacol       Date:  1995-09       Impact factor: 8.739

Review 6.  Safety of antihistamines in children.

Authors:  A P Ten Eick; J L Blumer; M D Reed
Journal:  Drug Saf       Date:  2001       Impact factor: 5.228
  6 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.