Literature DB >> 720385

Influence of GABA receptor agonists and antagonists on the binding of 3H-diazepam to the benzodiazepine receptor.

M S Briley, S Z Langer.   

Abstract

The GABA receptor agonists, GABA and muscimol, increased, while the GABA receptor antagonist, (+)-bicuculline, decreased the affinity of the benzodiazepine receptor for 3H-diazepam. The effect was seen at both 0 and 25 degrees C in spite of a large difference of affinity for 3H-diazepam at the two temperatures.

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Year:  1978        PMID： 720385     DOI： 10.1016/0014-2999(78)90031-6

Source DB:  PubMed          Journal:  Eur J Pharmacol        ISSN： 0014-2999            Impact factor:   4.432


  10 in total

Review 1.  Biochemical dissection of the gamma-aminobutyrate synapse.

Authors:  A J Turner; S R Whittle
Journal:  Biochem J       Date:  1983-01-01       Impact factor: 3.857

2.  Autoradiographic localization of benzodiazepine receptors in immunocytochemically identified gamma-aminobutyrergic synapses.

Authors:  H Möhler; J G Richards; J Y Wu
Journal:  Proc Natl Acad Sci U S A       Date:  1981-03       Impact factor: 11.205

3.  Proceedings of the British Pharmacological Society. University of Southampton, 17th-19th July 1985. Abstracts.

Authors: 
Journal:  Br J Pharmacol       Date:  1985-09       Impact factor: 8.739

4.  gamma-Aminobutyric acid and benzodiazepine receptors: copurification and characterization.

Authors:  M Gavish; S H Snyder
Journal:  Proc Natl Acad Sci U S A       Date:  1981-03       Impact factor: 11.205

5.  Anticonvulsant actions of the putative gamma-aminobutyric acid (GABA)-mimetic, ethylenediamine.

Authors:  P F Morgan; T W Stone
Journal:  Br J Pharmacol       Date:  1982-11       Impact factor: 8.739

Review 6.  The GABA postsynaptic membrane receptor-ionophore complex. Site of action of convulsant and anticonvulsant drugs.

Authors:  R W Olsen
Journal:  Mol Cell Biochem       Date:  1981-09-25       Impact factor: 3.396

7.  Effects of valproate on hyponeophagia in rats: competitive antagonism with picrotoxin and non-competitive antagonism with RO 15-1788.

Authors:  R A Shephard; D Stevenson; S Jenkinson
Journal:  Psychopharmacology (Berl)       Date:  1985       Impact factor: 4.530

8.  Pharmacological profile of the imidazopyridine zolpidem at benzodiazepine receptors and electrocorticogram in rats.

Authors:  S Arbilla; H Depoortere; P George; S Z Langer
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1985-09       Impact factor: 3.000

9.  Structure-activity studies on the potentiation of benzodiazepine receptor binding by ethylenediamine analogues and derivatives.

Authors:  P F Morgan; T W Stone
Journal:  Br J Pharmacol       Date:  1983-08       Impact factor: 8.739

10.  Methylmercury modulates GABAA receptor complex differentially in rat cortical and cerebellar membranes in vitro.

Authors:  H Komulainen; A Keränen; V Saano
Journal:  Neurochem Res       Date:  1995-06       Impact factor: 3.996
  10 in total

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