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1. CYP4F enzymes are the major enzymes in human liver microsomes that catalyze the O-demethylation of the antiparasitic prodrug DB289 [2,5-bis(4-amidinophenyl)furan-bis-O-methylamidoxime].

Authors: Michael Zhuo Wang; Janelle Y Saulter; Etsuko Usuki; Yen-Ling Cheung; Michael Hall; Arlene S Bridges; Greg Loewen; Oliver T Parkinson; Chad E Stephens; James L Allen; Darryl C Zeldin; David W Boykin; Richard R Tidwell; Andrew Parkinson; Mary F Paine; James Edwin Hall
Journal: Drug Metab Dispos Date: 2006-09-22 Impact factor: 3.922

2. Destruction of intracellular Trypanosoma cruzi after treatment of infected macrophages with cationic electron carriers.

Authors: M J Alves; M Rabinovitch
Journal: Infect Immun Date: 1983-01 Impact factor: 3.441

3. Enhanced permeability of the antimicrobial agent 2,5-bis(4-amidinophenyl)furan across Caco-2 cell monolayers via its methylamidoidme prodrug.

Authors: Liao Zhou; Kiho Lee; Dhiren R Thakker; David W Boykin; Richard R Tidwell; James E Hall
Journal: Pharm Res Date: 2002-11 Impact factor: 4.200

4. Synthesis of N-substituted aryl amidines by strong base activation of amines.

Authors: Muhammad M Khalifa; Micah J Bodner; J Andrew Berglund; Michael M Haley
Journal: Tetrahedron Lett Date: 2015-07-01 Impact factor: 2.415

5. Synthesis and antiprotozoal activity of cationic 1,4-diphenyl-1H-1,2,3-triazoles.

Authors: Stanislav A Bakunov; Svetlana M Bakunova; Tanja Wenzler; Maedot Ghebru; Karl A Werbovetz; Reto Brun; Richard R Tidwell
Journal: J Med Chem Date: 2010-01-14 Impact factor: 7.446

Review 6. Novel amidines and analogues as promising agents against intracellular parasites: a systematic review.

Authors: M N C Soeiro; K Werbovetz; D W Boykin; W D Wilson; M Z Wang; A Hemphill
Journal: Parasitology Date: 2013-04-08 Impact factor: 3.234

7. CYP1A1 and CYP1B1-mediated biotransformation of the antitrypanosomal methamidoxime prodrug DB844 forms novel metabolites through intramolecular rearrangement.

Authors: Wujian Ju; Sihyung Yang; John H Ansede; Chad E Stephens; Arlene S Bridges; Robert D Voyksner; Mohamed A Ismail; David W Boykin; Richard R Tidwell; James Edwin Hall; Michael Zhuo Wang
Journal: J Pharm Sci Date: 2013-11-01 Impact factor: 3.534

7 in total