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18 in total

1. A Back-to-Front Fragment-Based Drug Design Search Strategy Targeting the DFG-Out Pocket of Protein Tyrosine Kinases.

Authors: Hidehisa Iwata; Hideyuki Oki; Kengo Okada; Terufumi Takagi; Michiko Tawada; Yasushi Miyazaki; Shinichi Imamura; Akira Hori; J David Lawson; Mark S Hixon; Hiroyuki Kimura; Hiroshi Miki
Journal: ACS Med Chem Lett Date: 2012-02-28 Impact factor: 4.345

2. Alizarine derivatives as new dual inhibitors of the HIV-1 reverse transcriptase-associated DNA polymerase and RNase H activities effective also on the RNase H activity of non-nucleoside resistant reverse transcriptases.

Authors: Francesca Esposito; Tatyana Kharlamova; Simona Distinto; Luca Zinzula; Yung-Chi Cheng; Ginger Dutschman; Giovanni Floris; Patrick Markt; Angela Corona; Enzo Tramontano
Journal: FEBS J Date: 2011-03-16 Impact factor: 5.542

3. Alpha-retaining glucosyl transfer catalysed by trehalose phosphorylase from Schizophyllum commune: mechanistic evidence obtained from steady-state kinetic studies with substrate analogues and inhibitors.

Authors: B Nidetzky; C Eis
Journal: Biochem J Date: 2001-12-15 Impact factor: 3.857

4. Simple pseudo-dipeptides with a P2' glutamate: a novel inhibitor family of matrix metalloproteases and other metzincins.

Authors: Laurent Devel; Fabrice Beau; Mehdi Amoura; Laura Vera; Evelyne Cassar-Lajeunesse; Sandra Garcia; Bertrand Czarny; Enrico A Stura; Vincent Dive
Journal: J Biol Chem Date: 2012-06-11 Impact factor: 5.157

5. Substrate-binding recognition and specificity of trehalose phosphorylase from Schizophyllum commune examined in steady-state kinetic studies with deoxy and deoxyfluoro substrate analogues and inhibitors.

Authors: Christian Eis; Bernd Nidetzky
Journal: Biochem J Date: 2002-04-15 Impact factor: 3.857

6. Effects of DL-2-bromopalmitoyl-CoA and bromoacetyl-CoA in rat liver and heart mitochondria. Inhibition of carnitine palmitoyltransferase and displacement of [14C]malonyl-CoA from mitochondrial binding sites.

Authors: M R Edwards; M I Bird; E D Saggerson
Journal: Biochem J Date: 1985-08-15 Impact factor: 3.857

7. Interactions of nicotinamide-adenine dinucleotide phosphate analogues and fragments with pigeon liver malic enzyme. Synergistic effect between the nicotinamide and adenine moieties.

Authors: H J Lee; G G Chang
Journal: Biochem J Date: 1987-07-15 Impact factor: 3.857

8. Vinylogous ureas as a novel class of inhibitors of reverse transcriptase-associated ribonuclease H activity.

Authors: Michaela Wendeler; Hsiu-Fang Lee; Alun Bermingham; Jennifer T Miller; Oleg Chertov; Marion K Bona; Noel S Baichoo; Maryam Ehteshami; John Beutler; Barry R O'Keefe; Matthias Götte; Mamuka Kvaratskhelia; Stuart Le Grice
Journal: ACS Chem Biol Date: 2008-10-03 Impact factor: 5.100

9. Examination of α-exosite inhibitors against Botulinum neurotoxin A protease through structure-activity relationship studies of chicoric acid.

Authors: Song Xue; Hajime Seki; Marek Remes; Peter Šilhár; Kim Janda
Journal: Bioorg Med Chem Lett Date: 2017-10-12 Impact factor: 2.823

10. Exploiting drug-resistant enzymes as tools to identify thienopyrimidinone inhibitors of human immunodeficiency virus reverse transcriptase-associated ribonuclease H.

Authors: Takashi Masaoka; Suhman Chung; Pierluigi Caboni; Jason W Rausch; Jennifer A Wilson; Humeyra Taskent-Sezgin; John A Beutler; Graziella Tocco; Stuart F J Le Grice
Journal: J Med Chem Date: 2013-06-20 Impact factor: 7.446