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37 in total

1. Synthesis and structure-activity relationships of novel lincomycin derivatives. Part 2. Synthesis of 7(S)-7-deoxy-7-(4-morpholinocarbonylphenylthio)lincomycin and its 3-dimensional analysis with rRNA.

Authors: Yoshinari Wakiyama; Ko Kumura; Eijiro Umemura; Satomi Masaki; Kazutaka Ueda; Takashi Watanabe; Mikio Yamamoto; Yoko Hirai; Keiichi Ajito
Journal: J Antibiot (Tokyo) Date: 2015-12-16 Impact factor: 2.649

Review 2. New directions for macrolide antibiotics: structural modifications and in vitro activity.

Authors: H A Kirst; G D Sides
Journal: Antimicrob Agents Chemother Date: 1989-09 Impact factor: 5.191

3. Efficacy of cethromycin, a new ketolide, against Streptococcus pneumoniae susceptible or resistant to erythromycin in a murine pneumonia model.

Authors: E Azoulay-Dupuis; J Mohler; J P Bédos; C Barau; B Fantin
Journal: Antimicrob Agents Chemother Date: 2006-09 Impact factor: 5.191

4. In vitro activity and in vivo efficacy of a new series of 9-deoxo-12-deoxy-9,12-epoxyerythromycin A derivatives.

Authors: D J Hardy; R N Swanson; N L Shipkowitz; L A Freiberg; P A Lartey; J J Clement
Journal: Antimicrob Agents Chemother Date: 1991-05 Impact factor: 5.191

5. Synthesis and SARs of novel lincomycin derivatives Part 5: optimization of lincomycin analogs exhibiting potent antibacterial activities by chemical modification at the 6- and 7-positions.

Authors: Yoshinari Wakiyama; Ko Kumura; Eijiro Umemura; Satomi Masaki; Kazutaka Ueda; Yasuo Sato; Yoko Hirai; Yoshio Hayashi; Keiichi Ajito
Journal: J Antibiot (Tokyo) Date: 2017-11-01 Impact factor: 2.649

Chemical modification of erythromycins. I. Synthesis and antibacterial activity of 6-O-methylerythromycins A.

1. Synthesis and structure-activity relationships of novel lincomycin derivatives. Part 2. Synthesis of 7(S)-7-deoxy-7-(4-morpholinocarbonylphenylthio)lincomycin and its 3-dimensional analysis with rRNA.

Review 2. New directions for macrolide antibiotics: structural modifications and in vitro activity.

3. Efficacy of cethromycin, a new ketolide, against Streptococcus pneumoniae susceptible or resistant to erythromycin in a murine pneumonia model.

4. In vitro activity and in vivo efficacy of a new series of 9-deoxo-12-deoxy-9,12-epoxyerythromycin A derivatives.

5. Synthesis and SARs of novel lincomycin derivatives Part 5: optimization of lincomycin analogs exhibiting potent antibacterial activities by chemical modification at the 6- and 7-positions.

Review 6. Natural Products in the "Marketplace": Interfacing Synthesis and Biology.

Review 7. The macrolide antibiotic renaissance.

8. Isolation of a novel morphinan 3-O-diglucuronide metabolite from dog urine.

9. Synthesis and antibacterial activity of novel lincomycin derivatives. IV. Optimization of an N-6 substituent.

Review 10. The evolving role of chemical synthesis in antibacterial drug discovery.