Literature DB >> 6281658

Dimeric tetrapeptide enkephalins display extraordinary selectivity for the delta opiate receptor.

Y Shimohigashi, T Costa, H C Chen, D Rodbard.   

Abstract

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Year:  1982        PMID: 6281658     DOI: 10.1038/297333a0

Source DB:  PubMed          Journal:  Nature        ISSN: 0028-0836            Impact factor:   49.962


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  15 in total

1.  New potent biphalin analogues containing p-fluoro-L-phenylalanine at the 4,4' positions and non-hydrazine linkers.

Authors:  Adriano Mollica; Francesco Pinnen; Federica Feliciani; Azzurra Stefanucci; Gino Lucente; Peg Davis; Frank Porreca; Shou-Wu Ma; Josephine Lai; Victor J Hruby
Journal:  Amino Acids       Date:  2010-10-06       Impact factor: 3.520

2.  The effects of long-term treatment of NG108-15 cells with penta- and tetrapeptide enkephalin dimers on opioid receptor binding and cyclic AMP (cAMP) levels.

Authors:  S A Krumins
Journal:  Cell Mol Neurobiol       Date:  1987-06       Impact factor: 5.046

3.  A molecular dynamics study on opioid activities of biphalin molecule.

Authors:  Jin-Yuan Hsieh; Tzen-Yuh Chiang; Jun-Liang Chen; Yun-Wen Chen; Hong-Chang Lin; Chi-Chuan Hwang
Journal:  J Mol Model       Date:  2010-12-23       Impact factor: 1.810

4.  Design and synthesis of novel hydrazide-linked bifunctional peptides as delta/mu opioid receptor agonists and CCK-1/CCK-2 receptor antagonists.

Authors:  Yeon Sun Lee; Richard S Agnes; Hamid Badghisi; Peg Davis; Shou-wu Ma; Josephine Lai; Frank Porreca; Victor J Hruby
Journal:  J Med Chem       Date:  2006-03-09       Impact factor: 7.446

5.  A new opioid designed multiple ligand derived from the micro opioid agonist endomorphin-2 and the delta opioid antagonist pharmacophore Dmt-Tic.

Authors:  Severo Salvadori; Claudio Trapella; Stella Fiorini; Lucia Negri; Roberta Lattanzi; Sharon D Bryant; Yunden Jinsmaa; Lawrence H Lazarus; Gianfranco Balboni
Journal:  Bioorg Med Chem       Date:  2007-08-29       Impact factor: 3.641

6.  Solution-phase-peptide synthesis via the group-assisted purification (GAP) chemistry without using chromatography and recrystallization.

Authors:  Jianbin Wu; Guanghui An; Siqi Lin; Jianbo Xie; Wei Zhou; Hao Sun; Yi Pan; Guigen Li
Journal:  Chem Commun (Camb)       Date:  2014-02-07       Impact factor: 6.222

7.  Opioid-induced tolerance and dependence in mice is modulated by the distance between pharmacophores in a bivalent ligand series.

Authors:  David J Daniels; Natalie R Lenard; Chris L Etienne; Ping-Yee Law; Sandra C Roerig; Philip S Portoghese
Journal:  Proc Natl Acad Sci U S A       Date:  2005-12-19       Impact factor: 11.205

8.  Biological active analogues of the opioid peptide biphalin: mixed α/β(3)-peptides.

Authors:  Adriano Mollica; Francesco Pinnen; Roberto Costante; Marcello Locatelli; Azzurra Stefanucci; Stefano Pieretti; Peg Davis; Josephine Lai; David Rankin; Frank Porreca; Victor J Hruby
Journal:  J Med Chem       Date:  2013-04-12       Impact factor: 7.446

9.  Hydrazone Linker as a Useful Tool for Preparing Chimeric Peptide/Nonpeptide Bifunctional Compounds.

Authors:  Jolanta Dyniewicz; Piotr F J Lipiński; Piotr Kosson; Anna Leśniak; Marta Bochyńska-Czyż; Adriana Muchowska; Dirk Tourwé; Steven Ballet; Aleksandra Misicka; Andrzej W Lipkowski
Journal:  ACS Med Chem Lett       Date:  2016-11-01       Impact factor: 4.345

10.  Selectivities of opioid peptide analogues as agonists and antagonists at the delta-receptor.

Authors:  A D Corbett; M G Gillan; H W Kosterlitz; A T McKnight; S J Paterson; L E Robson
Journal:  Br J Pharmacol       Date:  1984-09       Impact factor: 8.739

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