Literature DB >> 6276785

[125I]-HEAT, a selective, high-affinity, high specific activity ligand for alpha 1-adrenoceptors.

H Glossmann, F Lübbecke, P Bellemann.   

Abstract

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Year:  1981        PMID： 6276785     DOI： 10.1007/bf00503304

Source DB:  PubMed          Journal:  Naunyn Schmiedebergs Arch Pharmacol        ISSN： 0028-1298            Impact factor:   3.000


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  12 in total

1.  Alpha noradrenergic receptors in brain membranes: sodium, magnesium and guanyl nucleotides modulate agonist binding.

Authors:  H Glossmann; P Presek
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1979-01       Impact factor: 3.000

2.  Solubilization of a mammalian beta-adrenergic receptor.

Authors:  J Kleinstein; H Glossmann; L Braun; C Konrad
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1978-12       Impact factor: 3.000

3.  [On the pharmacology of the alpha-receptor blocker BE 2254 (HEAT) (author's transl)].

Authors:  N Heinz; E Hofferber
Journal:  Arzneimittelforschung       Date:  1980

4.  Preferential blockade of postsynaptic alpha-adrenoceptors by BE 2254.

Authors:  M Göthert; J Nolte; G Weinheimer
Journal:  Eur J Pharmacol       Date:  1981-03-05       Impact factor: 4.432

Review 5.  Alpha-adrenoceptor subclassification.

Authors:  K Starke
Journal:  Rev Physiol Biochem Pharmacol       Date:  1981       Impact factor: 5.545

6.  Alpha 2 adrenoceptors in rat brain: the divalent cation site.

Authors:  H Glossmann; R Hornung
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1980-11       Impact factor: 3.000

7.  Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction.

Authors:  Y Cheng; W H Prusoff
Journal:  Biochem Pharmacol       Date:  1973-12-01       Impact factor: 5.858

8.  Cation sensitivity of [125I]heat binding to alpha 1-adrenoceptors in rat cerebral cortex membranes.

Authors:  H Glossmann; F Lübbecke; P Bellemann; P Presek
Journal:  Eur J Pharmacol       Date:  1981-10-22       Impact factor: 4.432

9.  Alpha adrenoceptors in rat brain: direct identification with prazosin.

Authors:  R Hornung; P Presek; H Glossmann
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1979-09       Impact factor: 3.000

10.  [125I]BE 2254, a new high affinity radioligand for alpha 1-adrenoceptors.

Authors:  G Engel; D Hoyer
Journal:  Eur J Pharmacol       Date:  1981-07-17       Impact factor: 4.432
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  5 in total

1.  Pharmacokinetic and alpha 1-adrenoceptor antagonistic properties of two cyanine-type inhibitors of extraneuronal monoamine transport.

Authors:  H Russ; B Friedgen; B Königs; C Schumacher; K H Graefe; E Schömig
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1996 Aug-Sep       Impact factor: 3.000

2.  Relationship between alpha 1-adrenoceptor density and functional response of rat vas deferens. Studies with phenoxybenzamine.

Authors:  K P Minneman; P W Abel
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1984-09       Impact factor: 3.000

3.  [125I]-HEAT:fifty percent of the ligand can bind to the alpha1-adrenoceptors with extremely high affinity.

Authors:  H Glossmann; F Lübbecke
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1982-10       Impact factor: 3.000

4.  [3H]ketanserin labels 5-HT2 receptors and alpha 1-adrenoceptors in human and pig brain membranes.

Authors:  D Hoyer; P Vos; A Closse; A Pazos; J M Palacios; H Davies
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1987-03       Impact factor: 3.000

5.  Radiation inactivation of alpha 1-adrenoceptors.

Authors:  F Lübbecke; D R Ferry; H Glossmann; E L Sattler; G Doell
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1983-06       Impact factor: 3.000
  5 in total

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