Literature DB >> 6270588

A steroid derivative, R 5135, antagonizes the GABA/benzodiazepine receptor interaction.

P Hunt, S Clements-Jewery.   

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Year:  1981        PMID: 6270588     DOI: 10.1016/0028-3908(81)90009-5

Source DB:  PubMed          Journal:  Neuropharmacology        ISSN: 0028-3908            Impact factor:   5.250


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  14 in total

1.  Clozapine and some other antipsychotic drugs may preferentially block the same subset of GABA(A) receptors.

Authors:  R F Squires; E Saederup
Journal:  Neurochem Res       Date:  1997-02       Impact factor: 3.996

2.  An electrophysiological investigation of the characteristics and function of GABAA receptors on bovine adrenomedullary chromaffin cells.

Authors:  J A Peters; J J Lambert; G A Cottrell
Journal:  Pflugers Arch       Date:  1989-10       Impact factor: 3.657

3.  An arylaminopyridazine derivative of gamma-aminobutyric acid (GABA) is a selective and competitive antagonist at the GABAA receptor site.

Authors:  J P Chambon; P Feltz; M Heaulme; S Restle; R Schlichter; K Biziere; C G Wermuth
Journal:  Proc Natl Acad Sci U S A       Date:  1985-03       Impact factor: 11.205

4.  Biphasic modulation of GABA(A) receptor binding by steroids suggests functional correlates.

Authors:  S Srinivasan; D W Sapp; A J Tobin; R W Olsen
Journal:  Neurochem Res       Date:  1999-11       Impact factor: 3.996

5.  Clozapine's antipsychotic effects do not depend on blockade of 5-HT3 receptors.

Authors:  R F Squires; E Saederup
Journal:  Neurochem Res       Date:  1999-05       Impact factor: 3.996

Review 6.  The diversity of GABAA receptors. Pharmacological and electrophysiological properties of GABAA channel subtypes.

Authors:  W Hevers; H Lüddens
Journal:  Mol Neurobiol       Date:  1998-08       Impact factor: 5.590

Review 7.  Advantages of an antagonist: bicuculline and other GABA antagonists.

Authors:  Graham A R Johnston
Journal:  Br J Pharmacol       Date:  2013-05       Impact factor: 8.739

8.  Clozapine and several other antipsychotic/antidepressant drugs preferentially block the same 'core' fraction of GABA(A) receptors.

Authors:  R F Squires; E Saederup
Journal:  Neurochem Res       Date:  1998-10       Impact factor: 3.996

9.  Beta-carboline binding indicates the presence of benzodiazepine receptor subclasses in the bovine central nervous system.

Authors:  K J Fehske; I Zube; H O Borbe; U Wollert; W E Müller
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1982-05       Impact factor: 3.000

10.  Antagonism of inhibitory amino acids by the steroid derivative RU5135.

Authors:  M A Simmonds; J P Turner
Journal:  Br J Pharmacol       Date:  1985-03       Impact factor: 8.739

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