Literature DB >> 6267448

Alternative explanation for the apparent "two-step" binding kinetics of high-affinity racemic antagonist radioligands.

E Bürgisser, R J Lefkowitz, A DeLean.   

Abstract

Mesh：

Substances：

Year:  1981        PMID： 6267448

Source DB:  PubMed          Journal:  Mol Pharmacol        ISSN： 0026-895X            Impact factor:   4.436


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  9 in total

1.  Experimental design and estimation of parameters in complex radioligand binding systems.

Authors:  C M Staschen; L D Homer
Journal:  J Pharmacokinet Biopharm       Date:  1996-12

2.  Properties of agonist binding at the beta-adrenoceptor of the rat reticulocyte.

Authors:  G Wiemer; A Wellstein; D Palm; H M von Hattingberg; D Brockmeier
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1982-10       Impact factor: 3.000

3.  Binding characteristics of (+)-, (+/-)- and (-)-[125iodo] cyanopindolol to guinea-pig left ventricle membranes.

Authors:  D Hoyer; G Engel; R Berthold
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1982-03       Impact factor: 3.000

4.  Ligand entry and exit pathways in the beta2-adrenergic receptor.

Authors:  Ting Wang; Yong Duan
Journal:  J Mol Biol       Date:  2009-08-06       Impact factor: 5.469

5.  Competitive and non-competitive interactions between specific ligands and beta-adrenoceptors in living cardiac cells.

Authors:  H Porzig; C Becker; H Reuter
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1982-11       Impact factor: 3.000

6.  [125I]-HEAT:fifty percent of the ligand can bind to the alpha1-adrenoceptors with extremely high affinity.

Authors:  H Glossmann; F Lübbecke
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1982-10       Impact factor: 3.000

7.  Recovery of beta-adrenoceptors and cyclic AMP response after long term treatment of intact heart cells with beta-blockers.

Authors:  C Becker; H Porzig
Journal:  Br J Pharmacol       Date:  1984-07       Impact factor: 8.739

8.  Binding of N-methylscopolamine to the extracellular domain of muscarinic acetylcholine receptors.

Authors:  Jan Jakubík; Alena Randáková; Pavel Zimčík; Esam E El-Fakahany; Vladimír Doležal
Journal:  Sci Rep       Date:  2017-01-16       Impact factor: 4.379

Review 9.  Binding kinetics of ligands acting at GPCRs.

Authors:  David A Sykes; Leigh A Stoddart; Laura E Kilpatrick; Stephen J Hill
Journal:  Mol Cell Endocrinol       Date:  2019-02-08       Impact factor: 4.102
  9 in total

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