Literature DB >> 6152826

The effect of sulphydryl block on the binding of H1-antagonists to the muscarinic receptor.

A S Burgen, C J Harbird.   

Abstract

The treatment of brain muscarinic receptors by p-chlormercuribenzoate is known to change structure-activity relationships for antagonists. The changes in binding affinity of H1-antagonists for this receptor have been measured; the changes are similar to those for intrinsic muscarinic antagonists.

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Year:  1983        PMID： 6152826      PMCID： PMC2045059          DOI： 10.1111/j.1476-5381.1983.tb10048.x

Source DB:  PubMed          Journal:  Br J Pharmacol        ISSN： 0007-1188            Impact factor:   8.739


  3 in total

1.  Heterogeneity of histamine H1-receptors: species variations in [3H]mepyramine binding of brain membranes.

Authors:  R S Chang; V T Tran; S H Snyder
Journal:  J Neurochem       Date:  1979-06       Impact factor: 5.372

2.  The effects of p-chloromercuribenzoate on muscarinic receptors in the cerebral cortex.

Authors:  N J Birdsall; A S Burgen; E C Hulme; E H Wong
Journal:  Br J Pharmacol       Date:  1983-09       Impact factor: 8.739

3.  The effect of p-chloromercuribenzoate on structure-binding relationships of muscarinic receptors in the rat cerebral cortex.

Authors:  N J Birdsall; A S Burgen; E C Hulme; E H Wong
Journal:  Br J Pharmacol       Date:  1983-09       Impact factor: 8.739
  3 in total

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