Literature DB >> 6140944

Chemical structure and biological activity of the diazepines.

P Danneberg, K H Weber.   

Abstract

Since the introduction of chlordiazepoxide and diazepam many diazepines have been developed. Use of these drugs is increasing and considerable knowledge has accumulated about their mechanisms of action. The structural and pharmacological properties of these drugs are surveyed briefly.

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Year:  1983        PMID： 6140944      PMCID： PMC1428206          DOI： 10.1111/j.1365-2125.1983.tb02295.x

Source DB:  PubMed          Journal:  Br J Clin Pharmacol        ISSN： 0306-5251            Impact factor:   4.335


  53 in total

1.  In vitro and in vivo inhibition by zopiclone of benzodiazepine binding to rodent brain receptors.

Authors:  J C Blanchard; A Boireau; C Garret; L Julou
Journal:  Life Sci       Date:  1979-06-25       Impact factor: 5.037

Review 2.  Effect of sedatives and anxiolytics on aggressivity.

Authors:  L Valzelli
Journal:  Mod Probl Pharmacopsychiatry       Date:  1979

3.  Benzodiazepines: potentiation of a GABA inhibitory response in the dorsal raphe nucleus.

Authors:  D W Gallager
Journal:  Eur J Pharmacol       Date:  1978-05-15       Impact factor: 4.432

4.  Increase of "antianxiety" activity and tolerance of behavioral depression during chronic administration of oxazepam.

Authors:  D L Margules; L Stein
Journal:  Psychopharmacologia       Date:  1968

5.  Benzodiazepine receptor: photoaffinity labeling and localization.

Authors:  M K Battersby; J G Richards; H Möhler
Journal:  Eur J Pharmacol       Date:  1979-08-01       Impact factor: 4.432

6.  A comparative study of certain pharmacologic responses following acute and chronic administrations of chlordiazepoxide.

Authors:  M E Goldberg; A A Manian; D H Efron
Journal:  Life Sci       Date:  1967-03-01       Impact factor: 5.037

7.  Benzodiazepine receptor-mediated experimental "anxiety" in primates.

Authors:  P T Ninan; T M Insel; R M Cohen; J M Cook; P Skolnick; S M Paul
Journal:  Science       Date:  1982-12-24       Impact factor: 47.728

8.  Ethyl beta-carboline-3-carboxylate shows differential benzodiazepine receptor interaction.

Authors:  M Nielsen; C Braestrup
Journal:  Nature       Date:  1980-08-07       Impact factor: 49.962

9.  The effect of central stimulant drugs on acetylcholine release from rat cerebral cortex.

Authors:  B A Hemsworth; M J Neal
Journal:  Br J Pharmacol       Date:  1968-11       Impact factor: 8.739

10.  Selective antagonists of benzodiazepines.

Authors:  W Hunkeler; H Möhler; L Pieri; P Polc; E P Bonetti; R Cumin; R Schaffner; W Haefely
Journal:  Nature       Date:  1981-04-09       Impact factor: 49.962
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  6 in total

1.  The use of vascular access ports for blood collection in feline blood donors.

Authors:  Isabelle Aubert; Anthony C G Abrams-Ogg; Anne M Sylvestre; Doris H Dyson; Dana G Allen; Ian B Johnstone
Journal:  Can J Vet Res       Date:  2011-01       Impact factor: 1.310

2.  The pharmacokinetics of clotiazepam after oral and sublingual administration to volunteers.

Authors:  C Benvenuti; V Bottà; M Broggini; V Gambaro; F Lodi; M Valenti
Journal:  Eur J Clin Pharmacol       Date:  1989       Impact factor: 2.953

3.  Anxiolytic-like profiles of histamine H3 receptor agonists in animal models of anxiety: a comparative study with antidepressants and benzodiazepine anxiolytic.

Authors:  Fumikazu Yokoyama; Miki Yamauchi; Masayo Oyama; Kunihiro Okuma; Kaname Onozawa; Takako Nagayama; Rie Shinei; Makoto Ishikawa; Yasuo Sato; Nobukazu Kakui
Journal:  Psychopharmacology (Berl)       Date:  2009-04-09       Impact factor: 4.530

4.  Synthesis and anticonvulsant activity of various mannich and schiff bases of 1,5-benzodiazepines.

Authors:  Surendra N Pandeya; Neha Rajput
Journal:  Int J Med Chem       Date:  2012-11-28

Review 5.  Review of withdrawal catatonia: what does this reveal about clozapine?

Authors:  Matthew Lander; Tarun Bastiampillai; Jitender Sareen
Journal:  Transl Psychiatry       Date:  2018-07-31       Impact factor: 6.222

6.  Synthesis and Anti-Proliferative Assessment of Triazolo-Thiadiazepine and Triazolo-Thiadiazine Scaffolds.

Authors:  Ahmed T A Boraei; Hazem A Ghabbour; Mohamed S Gomaa; El Sayed H El Ashry; Assem Barakat
Journal:  Molecules       Date:  2019-12-06       Impact factor: 4.411
  6 in total

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