Literature DB >> 6118436

gamma-Aminobutyric acid agonists, antagonists, and uptake inhibitors. Design and therapeutic aspects.

P Krogsgaard-Larsen.   

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Year:  1981        PMID： 6118436     DOI： 10.1021/jm00144a001

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  7 in total

1.  An arylaminopyridazine derivative of gamma-aminobutyric acid (GABA) is a selective and competitive antagonist at the GABAA receptor site.

Authors:  J P Chambon; P Feltz; M Heaulme; S Restle; R Schlichter; K Biziere; C G Wermuth
Journal:  Proc Natl Acad Sci U S A       Date:  1985-03       Impact factor: 11.205

Review 2.  Molecular biology of inhibitory amino acid receptors.

Authors:  R S Duman; P M Sweetnam; P A Gallombardo; J F Tallman
Journal:  Mol Neurobiol       Date:  1987 Spring-Summer       Impact factor: 5.590

3.  Ligand-binding studies on GABA receptors--relation to physiology and behavior.

Authors:  F V DeFeudis
Journal:  Neurochem Res       Date:  1984-03       Impact factor: 3.996

4.  Vigabatrin transport across the human intestinal epithelial (Caco-2) brush-border membrane is via the H+ -coupled amino-acid transporter hPAT1.

Authors:  Emily L Abbot; Danielle S Grenade; David J Kennedy; Kelly M Gatfield; David T Thwaites
Journal:  Br J Pharmacol       Date:  2006-02       Impact factor: 8.739

5.  GABA receptors on the somatic muscle cells of the parasitic nematode, Ascaris suum: stereoselectivity indicates similarity to a GABAA-type agonist recognition site.

Authors:  L Holden-Dye; P Krogsgaard-Larsen; L Nielsen; R J Walker
Journal:  Br J Pharmacol       Date:  1989-11       Impact factor: 8.739

6.  Synthesis and evaluation of novel aromatic substrates and competitive inhibitors of GABA aminotransferase.

Authors:  Michael D Clift; Richard B Silverman
Journal:  Bioorg Med Chem Lett       Date:  2007-10-22       Impact factor: 2.823

7.  Retinal Electrophysiology Is a Viable Preclinical Biomarker for Drug Penetrance into the Central Nervous System.

Authors:  Jason Charng; Zheng He; Algis J Vingrys; Rebecca L Fish; Rachel Gurrell; Bang V Bui; Christine T Nguyen
Journal:  J Ophthalmol       Date:  2016-04-27       Impact factor: 1.909
  7 in total

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