Literature DB >> 590345

3H-Spiroperidol labels dopamine receptors in pituitary and brain.

I Creese, R Schneider, S H Snyder.   

Abstract

3H-Spiroperidol of high specific radioactivity labels dopamine receptors in membranes of bovine caudate nucleus and anterior pituitary. The saturation and kinetic properties of 3H-spiroperidol binding are similar in the two tissues. In both caudate and pituitary 3H-spiroperidol displays very high affinity with a dissociation constant of 0.2-0.3 nM. The relative potencies of numerous dopamine agonists and antagonists in competing for 3H-spiroperidol binding are closely similar in anterior pituitary and caudate.

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Year:  1977        PMID： 590345     DOI： 10.1016/0014-2999(77)90232-1

Source DB:  PubMed          Journal:  Eur J Pharmacol        ISSN： 0014-2999            Impact factor:   4.432


  40 in total

1.  Sensitivity of morphine-tolerant rats to muscarinic and dopaminergic agonists: relation to tolerance or withdrawal.

Authors:  M J Christie; D H Overstreet
Journal:  Psychopharmacology (Berl)       Date:  1979-09       Impact factor: 4.530

Review 2.  Control of prolactin secretion by excitatory amino acids.

Authors:  György M Nagy; Ibolya Bodnár; Zsuzsanna Bánky; Béla Halász
Journal:  Endocrine       Date:  2005-12       Impact factor: 3.633

3.  Differential response of central dopaminergic system in acute and chronic unpredictable stress models in rats.

Authors:  Naila Rasheed; Ausaf Ahmad; Chandra Prakash Pandey; Rajnish Kumar Chaturvedi; Mohtashim Lohani; Gautam Palit
Journal:  Neurochem Res       Date:  2009-07-01       Impact factor: 3.996

4.  Subsensitivity of the rat striatal dopaminergic system after treatment with bromocriptine: effects on [3H]spiperone binding and dopamine-stimulated cyclic AMP formation.

Authors:  M Quik; L L Iversen
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1978-09       Impact factor: 3.000

5.  Effects of ceruletide on the dopamine receptor-adenylate cyclase system in striatum and frontal cortex of rats chronically treated with haloperidol.

Authors:  Y Hatta; S Hatta; T Saito
Journal:  Psychopharmacology (Berl)       Date:  1993       Impact factor: 4.530

6.  Elucidation of the structure and receptor binding studies of the major primary, metabolite of dihydroergotamine in man.

Authors:  G Maurer; W Frick
Journal:  Eur J Clin Pharmacol       Date:  1984       Impact factor: 2.953

7.  Dopamine receptors in canine caudate nucleus.

Authors:  H Maeno
Journal:  Mol Cell Biochem       Date:  1982-03-19       Impact factor: 3.396

8.  Effects of ceruletide on perioral movements and the dopamine receptor-adenylate cyclase system in rats chronically treated with fluphenazine.

Authors:  T Ashizawa; T Saito; N Takahata
Journal:  Psychopharmacology (Berl)       Date:  1996-06       Impact factor: 4.530

9.  Differential reversal of various dopamine antagonists by anticholinergics in Sidman avoidance: possible relationship to adrenergic blockade.

Authors:  J M Liebman; R Neale; L Noreika; A Braunwalder
Journal:  Psychopharmacology (Berl)       Date:  1981       Impact factor: 4.530

10.  Receptor inhibition by immunoglobulins: specific inhibition by autistic children, their relatives, and control subjects.

Authors:  E H Cook; B D Perry; G Dawson; M S Wainwright; B L Leventhal
Journal:  J Autism Dev Disord       Date:  1993-03
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