Literature DB >> 5677227

1-acyl-indoles. II. A new syntheses of 1-(p-chlorobenzoyl)-5-methyoxy-3-indolyacetic acid and its polymorphism.

H Yamamoto.   

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Year:  1968        PMID： 5677227     DOI： 10.1248/cpb.16.17

Source DB:  PubMed          Journal:  Chem Pharm Bull (Tokyo)        ISSN： 0009-2363            Impact factor:   1.645


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  12 in total

1.  Indomethacin Analogues that Enhance Doxorubicin Cytotoxicity in Multidrug Resistant Cells without Cox Inhibitory Activity.

Authors:  Mitsuhiro Arisawa; Yayoi Kasaya; Tohru Obata; Takuma Sasaki; Mika Ito; Hiroshi Abe; Yoshihiro Ito; Akihito Yamano; Satoshi Shuto
Journal:  ACS Med Chem Lett       Date:  2011-03-17       Impact factor: 4.345

2.  A kinetic study of the polymorphic transformation of nimodipine and indomethacin during high shear granulation.

Authors:  Zhen Guo; Mingxin Ma; Tianyi Wang; Di Chang; Tongying Jiang; Siling Wang
Journal:  AAPS PharmSciTech       Date:  2011-05-07       Impact factor: 3.246

3.  Spectroscopic characterization of interactions between PVP and indomethacin in amorphous molecular dispersions.

Authors:  L S Taylor; G Zografi
Journal:  Pharm Res       Date:  1997-12       Impact factor: 4.200

4.  Solid-state characteristics of amorphous sodium indomethacin relative to its free acid.

Authors:  P Tong; G Zografi
Journal:  Pharm Res       Date:  1999-08       Impact factor: 4.200

5.  Straightforward protocol for the efficient synthesis of varied N(1)-acylated (aza)indole 2-/3-alkanoic acids and esters: optimization and scale-up.

Authors:  Andy J Liedtke; Kwangho Kim; Donald F Stec; Gary A Sulikowski; Lawrence J Marnett
Journal:  Tetrahedron       Date:  2012-12-02       Impact factor: 2.457

Review 6.  Aldo-Keto Reductase (AKR) 1C3 inhibitors: a patent review.

Authors:  Trevor M Penning
Journal:  Expert Opin Ther Pat       Date:  2017-09-19       Impact factor: 6.674

7.  Synthesis and investigations of double-pharmacophore ligands for treatment of chronic and neuropathic pain.

Authors:  Ruben Vardanyan; Gokhale Vijay; Gary S Nichol; Lu Liu; Isuru Kumarasinghe; Peg Davis; Todd Vanderah; Frank Porreca; Josephine Lai; Victor J Hruby
Journal:  Bioorg Med Chem       Date:  2009-06-02       Impact factor: 3.641

8.  Polymorphic Transformation of Indomethacin during Hot Melt Extrusion Granulation: Process and Dissolution Control.

Authors:  Ting Xu; Kajalajit Nahar; Rutesh Dave; Simon Bates; Kenneth Morris
Journal:  Pharm Res       Date:  2018-05-10       Impact factor: 4.200

9.  Development of potent and selective indomethacin analogues for the inhibition of AKR1C3 (Type 5 17β-hydroxysteroid dehydrogenase/prostaglandin F synthase) in castrate-resistant prostate cancer.

Authors:  Andy J Liedtke; Adegoke O Adeniji; Mo Chen; Michael C Byrns; Yi Jin; David W Christianson; Lawrence J Marnett; Trevor M Penning
Journal:  J Med Chem       Date:  2013-03-13       Impact factor: 7.446

10.  Controlling Indomethacin Release through Vapor-Phase Deposited Hydrogel Films by Adjusting the Cross-linker Density.

Authors:  Paul Christian; Stephan Tumphart; Heike M A Ehmann; Hans Riegler; Anna Maria Coclite; Oliver Werzer
Journal:  Sci Rep       Date:  2018-05-08       Impact factor: 4.379
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